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3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]propan-1-one
7-(3-chlorophenyl)-4-[(4-hydroxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[(2S)-oxolane-2-carbonyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
7-(2-methoxyethyl)-2-(1-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-(ethylamino)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]pyrimidine-5-carboxamide
(1S,5R)-3-(1H-1,3-benzodiazole-5-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(3R,4S)-4-(4-methoxyphenyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-amine
4-(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}pyrrolidin-2-yl)-3,5-dimethyl-1,2-oxazole
2-{1-[(3-methoxyphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(1-acetylpiperidin-3-yl)methyl]-3-(4-methoxyphenyl)propanamide
3-(2,5-difluorobenzoyl)-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine
N-[1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
N-{[(3S,4S)-3-hydroxy-1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]methyl}cyclopentanecarboxamide
4-(2-methoxyethoxy)-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine
2-{1-[(3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[3-({ethyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]carbamoyl}amino)-4-methylphenyl]acetamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
(1R,2R,6S,7S)-4-(1H-indole-7-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1,3-trimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{[(2R,5S)-5-(pyridin-3-ylmethyl)oxolan-2-yl]methyl}thiomorpholine
1-[(5-fluoro-2-methoxyphenyl)methyl]-4-methoxypiperidine
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N,2,3-trimethylquinoxaline-6-carboxamide
1-(4-tert-butylphenyl)-3-[(5-methylpyrazin-2-yl)methyl]urea
1-ethyl-N,2,5-trimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrrole-3-carboxamide
1-methyl-4-(5-phenylpentanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(1-{7-[2-(dimethylamino)benzoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)methanesulfonamide
ethyl 1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)acetyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(1R,5S)-3-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3,8-diazabicyclo[3.2.1]octane
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
(3S,4S)-1-cyclohexyl-4-cyclopropylpyrrolidine-3-carboxylic acid
3-(5-methyl-1H-pyrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]propan-1-one
3-ethoxy-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-{1-[1-(cyclohexylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
(3S)-1-{5-[(3S)-3-ethylmorpholine-4-carbonyl]-1-methyl-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
(1S,5R)-3-(4-methylpyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 1-benzyl-5-[(2-methylpropyl)amino]-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-N-[2-(propan-2-yloxy)ethyl]piperidine-4-carboxamide
4-hydroxy-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-2-(phenoxymethyl)pyrimidine-5-carboxamide
N-cyclopropyl-3-[1-(5-phenylpentanoyl)piperidin-4-yl]propanamide
6-methoxy-4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-{4-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]phenyl}ethan-1-one
N-benzyl-1-(2-hydroxyethyl)-5-[4-(4-methoxyphenyl)butan-2-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
1-{2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-3-(1H-imidazol-1-ylmethyl)piperidine
5-methyl-3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}-1H-indazole
3-(2-methoxyphenyl)-N-[(3-methyloxetan-3-yl)methyl]propanamide
N-[2-(diethylamino)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methylbenzamide
N-[(2R,3R)-1'-(4-methyl-2-oxopentanoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide