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(2S,4R)-N-ethyl-1-[3-(methylsulfanyl)propyl]-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-ethyl-9-[(8-fluoroquinolin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-3-(pyridin-4-yl)propanamide
1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[2-(pyridin-3-yloxy)propyl]urea
1-methyl-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-acetyl-N-(1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-2-carboxamide
[1-(4-chloro-2,5-dimethylbenzenesulfonyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
1-{4-[(2,3-dihydroxypropyl)(methyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-methoxy-1-[4-(4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}phenoxy)piperidin-1-yl]ethan-1-one
1-cyclopentyl-5-oxo-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}pyrrolidine-3-carboxamide
2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
N-{1-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N,5-dimethyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
4-oxo-1-[2-(2-oxoimidazolidin-1-yl)ethyl]-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
methyl 4-[4-({4-[hydroxy(thiophen-2-yl)methyl]piperidin-1-yl}methyl)-5-methyl-1,3-oxazol-2-yl]benzoate
5-ethyl-1'-(2-methylquinolin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-{[1-(pyrazin-2-yl)piperidin-4-yl]methyl}benzoic acid
ethyl 5-{[(2H-1,3-benzodioxol-5-ylmethyl)amino]methyl}-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
4-{2-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-cyclohexyl-5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)-N-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
5-[1-(1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-methyl-4-(piperidin-3-ylmethyl)-N-(quinolin-5-ylmethyl)benzamide
3-(1-benzofuran-2-yl)-1-benzyl-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(5-phenyl-1,2-oxazole-3-carbonyl)piperazine
1-cyclopropanecarbonyl-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-4-carboxamide
3,4-difluoro-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)benzene-1-sulfonamide
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]ethan-1-one
1-(cyclopropylmethyl)-4-(2-methyl-1,3-thiazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-{2-[4-(6-methylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzene-1-sulfonamide
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-2-(pyrrolidin-1-ylmethyl)piperidine
3-{[1-(3-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
3-(4-methoxyphenyl)-1-{4-[2-(pyridin-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(thiomorpholin-4-yl)pyridine-3-carboxamide
2-methyl-1-(propan-2-yl)-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine
methyl (2S)-2-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamido}-3-phenylpropanoate
1-[4-(ethylsulfanyl)phenyl]-3-[2-(3-methoxyphenoxy)ethyl]-3-methylurea
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)ethan-1-one
5-(2-chlorophenyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]furan-2-carboxamide
3-{[4-(2,3-difluoro-6-methoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)propanamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-[3-(pyridine-3-carbonyl)piperidin-1-yl]ethan-1-one
(3S,7S)-5-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-triene-3-carboxylic acid
1-{1'-[5-(methoxymethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(1R,5R)-3-(2-chlorobenzenesulfonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-methoxyethyl)-1-methyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydroquinoline-3-carboxamide
5-(1H-indole-6-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[2-(propylsulfanyl)phenyl]-4-(1H-pyrazol-3-yl)piperidine-1-carboxamide
6-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one