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4-(6-cyclopropylpyrimidin-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-methoxy-N-methyl-2-phenyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-1,4-oxazepan-6-ol
3-fluoro-N-[(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
6-ethyl-3-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-1,5-dimethyl-1,2-dihydropyridin-2-one
2-[4-(1H-imidazol-1-yl)butanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(2S)-N-[4-(difluoromethoxy)-2-methylphenyl]-2-(morpholine-4-carbonyl)pyrrolidine-1-carboxamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-3-(thiophen-3-yl)propan-1-one
(1S,6R)-9-[(2,6-difluoro-3-methylphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
5-cyclopropanecarbonyl-1'-[(2-methoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-methyl-2,6-dioxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)(methyl)amino]methyl}-1-cyclopentylpyrrolidin-2-one
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
1-tert-butyl-3-methyl-5-[(3-methylphenyl)methyl]-1H-1,2,4-triazole
N'-[(4-ethylphenyl)methyl]-N'-(2-methoxyethyl)-N-(4-methyl-1,3-thiazol-2-yl)ethanediamide
2-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}benzoic acid
6-methyl-4-{2-oxo-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
6-ethyl-N-[1-(methoxymethyl)cyclopentyl]-2-methylquinoline-4-carboxamide
6-(2-fluorophenyl)-N-methyl-N-(oxan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
14-(1-ethyl-1H-1,2,4-triazol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
3-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
5-[2-(2-methoxyphenyl)acetyl]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-2-(morpholin-4-yl)acetamide
N-(adamantan-2-yl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-2-(trifluoromethyl)morpholine
(3S,5R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-N-[(5-methylfuran-2-yl)methyl]acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-2-one
3-(2-cyclopropyl-1,3-dioxo-2,3-dihydro-1H-isoindol-5-yl)-1-[1-(4-propyl-4H-1,2,4-triazol-3-yl)ethyl]urea
2-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-8-methyl-2,8-diazaspiro[5.5]undecane
5-[3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyrrolidin-2-one
{1-[2-(2-methylphenyl)benzoyl]-3-[(2-methylphenyl)methyl]piperidin-3-yl}methanol
(2S,4R)-4-amino-N-ethyl-1-[4-(2-methylfuran-3-amido)benzoyl]pyrrolidine-2-carboxamide
5-({[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}amino)-1-ethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
5-{1-[(2,3-dimethoxyphenyl)methyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
1-cyclobutanecarbonyl-4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1,4-diazepane
4-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-3-propyl-1H-pyrazole
(4aS,8aR)-1-(3-aminopropyl)-6-(2-chlorobenzoyl)-decahydro-1,6-naphthyridin-2-one
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
1-[3-(2-phenylethyl)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
(1S,5R)-N-(2,4-difluorophenyl)-6-(3-methylbut-2-en-1-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
methyl 5-{[(3-fluorophenyl)methyl]amino}-1-(2-methoxyethyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S)-1-(2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetyl)pyrrolidine-2-carboxylate
1-(2,6-dimethoxybenzoyl)-4-(4-fluorophenyl)-1,4-diazepane
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(pyridin-2-yl)acetamide
1-cyclopropyl-N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-5-oxopyrrolidine-3-carboxamide
1-(2-fluorobenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(1H-pyrazol-1-yl)benzamide