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(2S,4R)-N-(2-methyl-1,3-benzothiazol-5-yl)-1-(3-phenylpropyl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-5-methylpyridine-3-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[2-(morpholin-4-yl)ethyl]piperidine-3,5-dicarboxamide
(3S,4R)-3-benzyl-1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-methylpiperidin-4-ol
(1R,7S)-6-(4-fluoropiperidine-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
ethyl 1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
2-[(4aS,8aR)-4a-(hydroxymethyl)-1-[(5-methylfuran-2-yl)methyl]-decahydro-1,6-naphthyridin-6-yl]pyridine-3-carboxamide
4-[2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)ethyl]benzene-1-sulfonamide
methyl 2-hydroxy-5-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)benzoate
4-(4-methyl-2-phenylpyrimidine-5-carbonyl)-1,4-oxazepan-6-ol
N-(3,3-diphenylpropyl)-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-methyl-5-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}pyrazine
2-(2-aminoethyl)-N-[1-(thiophen-2-yl)propyl]quinazolin-4-amine
2-methyl-3-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}quinoxaline
4-(4-fluorophenyl)-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-ol
1-ethyl-3-methyl-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole
3-(1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-4-yl)-N-phenylpropanamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(6-methoxy-1H-indazol-3-yl)methyl]methylamine
[9-(1H-imidazol-2-ylmethyl)-3-(thiophen-3-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-{1-[(2-ethoxyphenyl)methyl]-4-[(6-methoxy-2H-chromen-3-yl)methyl]piperazin-2-yl}ethan-1-ol
6-fluoro-N-methyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(methanesulfonylmethyl)piperidine
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
4-methyl-2-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]phenol
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)imidazo[1,2-a]pyrimidine-2-carboxamide
N-[2-(pyridin-3-yloxy)ethyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
7a-({2-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1H-imidazol-1-yl}methyl)-hexahydro-1H-pyrrolizine
N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)hept-6-ynamide
4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]-1,4-oxazepane
2-methyl-4-{4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}pyridine
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
4-(2-amino-6-methylpyrimidin-4-yl)-3-methyl-1-phenylpiperazin-2-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2,1-benzoxazole-3-carboxamide
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-methyl-4-{[(2R,5S)-5-{[4-(trifluoromethoxy)phenyl]methyl}oxolan-2-yl]methyl}piperazine
1-[3-(3-ethylphenoxy)azetidin-1-yl]-3-[methyl(1-methylpyrrolidin-3-yl)amino]propan-1-one
ethyl 4-[(5S,9aS,9bS)-2-cyclopentyl-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]-1H-pyrazole-3-carboxylate
5-ethyl-5-[1-(6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[3-(5-methylfuran-2-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-{1-[1-(4-chlorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]urea
2,5-dimethyl-3-{4-[4-(pyridin-3-yl)pyrimidin-2-yl]piperazin-1-yl}pyrazine
4-(3-{1-[2-(morpholin-4-yl)ethyl]-1H-pyrazol-3-yl}phenyl)isoquinoline
1-(1-methyl-3-phenyl-1H-pyrazole-5-carbonyl)-2-[2-(pyrrolidin-1-yl)ethyl]piperidine
2-(butylsulfanyl)-6-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]pyrimidin-4-amine
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
N-cyclohexyl-3-[2-(2,3-difluoro-6-methoxyphenyl)-1H-imidazol-1-yl]propanamide
2-(methylsulfanyl)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one