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1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(3-methoxypropyl)benzamide
1-{4-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
4-{[1-(2-acetamidoacetyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-cyclopropanecarbonyl-1'-(4-methyl-1,3-thiazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-methoxy-N-{3-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]phenyl}benzamide
ethyl 4-[(4-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine-1-carboxylate
N-[(2,4-difluorophenyl)methyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-[(4-fluorophenyl)methyl]-N-methyl-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(2,3-dihydro-1H-inden-2-yl)-2-(1H-imidazol-4-yl)-1H-imidazole
2-{[(adamantan-1-yl)amino]methyl}-4-phenylphenol
N-({1-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}methyl)thiophene-2-carboxamide
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-[(1-benzylpiperidin-4-yl)methyl]-N,4-dimethylpyrimidine-5-carboxamide
ethyl 4-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine-1-carboxylate
ethyl 2-{1-[1-(2-methoxyethyl)-6-oxopiperidine-3-amido]cyclohexyl}acetate
N-cyclooctyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
3-methyl-1-(1-{6-[3-(1H-pyrazol-1-yl)azetidin-1-yl]pyridine-3-carbonyl}piperidin-3-yl)butan-1-one
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
2-amino-1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(2,3-dihydro-1H-inden-2-yl)piperidine
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
N-(2-methylphenyl)-N'-(4-phenylbutyl)propanediamide
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]pyrrolidin-2-yl}-N-(propan-2-yl)thiophene-2-carboxamide
(2S)-2-amino-3-(1H-indol-3-yl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
N-{1-[1-(2-chloropyridine-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-4-phenylbutanamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-propyl-1H-pyrazole-5-carboxamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1,8-naphthyridine-2-carboxamide
(1S,5R)-3-benzyl-6-(4-propylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,2-difluoroethyl)-4-{[2-(1H-imidazol-4-yl)ethyl]sulfamoyl}benzamide
methyl (2S,4R)-1-(1-benzylpiperidin-4-yl)-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
N-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2-methoxy-2-methylpropanamide
N-[(2R,3R)-1'-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(1,3-benzoxazol-2-yl)acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
4,5-dimethyl 1-[(3S,5S)-5-[(furan-2-ylmethyl)carbamoyl]-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
2-{[4-(4-amino-5-methylpyrimidin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}ethan-1-ol
N-methyl-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(5-fluoropyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2,4-dimethoxy-6-[3-(1H-pyrazol-3-yl)phenyl]-1,3,5-triazine
7-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxalin-2-one
3-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}pyridin-2-amine
N-(oxan-3-ylmethyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
methyl 3-benzamido-1-(oxolan-2-ylmethyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-[(1-phenylcyclopentyl)methyl]propanamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-3-methoxypropanamide
3-{[1-(4-chlorobenzoyl)pyrrolidin-3-yl]methyl}benzamide
1-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]-3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}propan-1-one