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N-ethyl-2-[2-(pyrimidin-2-ylsulfanyl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
2-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}pyridine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-1H-pyrrole-3-carboxamide
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(1H-pyrrol-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-({[3-(1,3-benzothiazol-2-yl)propyl]amino}methyl)pyrrolidin-3-ol
2-methoxy-N-[1-(2-phenylethyl)-7-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl]acetamide
5-({4-[(2-fluorophenyl)methyl]piperidin-1-yl}methyl)-N,N-dimethyl-1,3-thiazol-2-amine
3-(oxolan-2-ylmethyl)-5-[1-(1-phenylcyclopropanecarbonyl)piperidin-4-yl]-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
1-cyclohexyl-N3-(cyclopropylmethyl)-N5-methyl-4-oxo-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}urea
1-[4-(2-{[(furan-2-ylmethyl)(prop-2-yn-1-yl)amino]methyl}quinazolin-4-yl)piperazin-1-yl]ethan-1-one
3-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzonitrile
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(2-methylphenyl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-{4-[(3-phenoxyazetidin-1-yl)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
N4-(2H-1,3-benzodioxol-5-yl)-N2-(pyridin-2-ylmethyl)morpholine-2,4-dicarboxamide
4-(6-methylpyridazin-3-yl)-2,2-diphenylbutanenitrile
1-cyclopentyl-4-oxo-N-[(4-phenyloxan-4-yl)methyl]-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
{4-[4-(1H-pyrrol-1-yl)benzoyl]-1,4-oxazepan-6-yl}methanol
3-amino-2-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(4-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(thiophen-3-ylmethyl)amine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-4-(2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carbonyl)morpholine
(3R,5R)-N-[(2-ethoxypyridin-3-yl)methyl]-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}[1-(morpholin-4-yl)propan-2-yl]amine
3-methoxy-N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
1-[4-(difluoromethoxy)benzoyl]-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-methyl-1,4-diazepan-5-one
(4aS,8aR)-6-[(2-phenyl-1,3-oxazol-4-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-(1H-indol-3-yl)ethyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
9-(2,3-dihydro-1H-indene-1-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-1-(2,3,5-trifluorophenyl)urea
4-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine-3-carbonyl)pyridin-2-amine
1-[3-({[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]amino}methyl)pyridin-2-yl]piperidin-3-ol
2-{[1-(6-aminopyridin-3-yl)-4-methyl-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
ethyl 4-(7-{[2-(methoxycarbonyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidine-1-carboxylate
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
N-(5-chloro-2-methoxyphenyl)-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carboxamide
3-[(3R,4S)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-methoxy-N-[4-(2-methoxypyrimidin-5-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]acetamide
2,6-dihydroxy-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)benzamide
(1R,3S)-3-{[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(1,2-oxazole-3-carbonyl)piperidin-3-ol
5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-[3-(3-{[4-(2,3-dimethylphenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3,5-dimethoxybenzamide
5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-ethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-6-oxopiperidine-3-carboxamide
3-methyl-N-[(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}pyrrolidin-3-yl)methyl]furan-2-carboxamide
(2S,4S)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxylic acid