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2-{5-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}propanamide
4-(1-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}ethyl)morpholine
2-[(5-methylpyrazin-2-yl)methyl]-9-(2-phenoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-methylpiperidin-2-one
3-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
(4aS,8aS)-2-[(2-methoxypyrimidin-5-yl)methyl]-decahydroisoquinolin-4a-ol
(3S,4S)-3-hydroxy-4-(propan-2-yloxy)-N-(3,4,5-trimethoxyphenyl)pyrrolidine-1-carboxamide
1-(3-chloro-4-ethoxyphenyl)-3-(2-methoxyethyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
1-(4-chloro-2,6-dimethylphenyl)-3-(2-hydroxyethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]urea
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-[3-(4-methylphenyl)propanoyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
4-{2-methyl-6-[1-(morpholine-2-carbonyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
1-[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-triazin-3-yl]-4-phenylazepane
2-[4-(3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
ethyl 1-{[1-(hydroxymethyl)cyclobutyl]methyl}-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
3-methyl-1-[2-oxo-2-(2-phenylpyrrolidin-1-yl)ethyl]-1,2-dihydroquinoxalin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetamide
4-[(1-{3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}piperidin-3-yl)methyl]benzoic acid
ethyl 2-[1-(2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-2-yl]acetate
4-(1-methyl-1H-imidazol-2-yl)-1-(2-phenoxyethyl)-1H-1,2,3-triazole
4-(2,3-dimethylphenyl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
1-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]cyclopropane-1-carbonitrile
N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
4-({1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}methyl)benzoic acid
(1S,5R)-6-(2-methoxyethyl)-3-[4-(1H-pyrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
[(4-fluoro-3-methoxyphenyl)methyl](methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-(pyridin-4-ylmethyl)-9-(trimethylpyrimidin-4-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-({5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazol-3-yl}formamido)acetamide
5-(4-benzoylpiperazine-1-carbonyl)quinoxaline
4-(cyclohexylmethyl)-3-(4-hydroxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S)-N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-methylpentanamide
N-(1-{1-[2-(2,3,6-trifluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopropanecarboxamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-3-methylurea
2-(4-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-1-(2-phenylethyl)piperazin-2-yl)ethan-1-ol
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}urea
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(pyridin-4-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N4-[2-(1H-imidazol-1-yl)ethyl]-N2,N2,5,6-tetramethylpyrimidine-2,4-diamine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
2-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-3-carboxylic acid
2-[4-(1H-1,3-benzodiazol-1-yl)phenyl]-N-ethylacetamide
N-({3,5-dimethoxy-4-[2-(thiophen-3-yl)ethoxy]phenyl}methyl)-3-fluoro-N-[(3S)-2-oxoazepan-3-yl]benzamide
2-[(cyclopropylmethyl)sulfanyl]-1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
6-(4-ethenylbenzoyl)-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-({2-[(3-methoxyphenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
7-(cyclopropylmethyl)-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decane