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ethyl 4-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}piperazine-1-carboxylate
3-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5-[4-(trifluoromethyl)phenyl]-1,2,4-triazine
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
N-[(2-fluorophenyl)methyl]-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]propanamide
1-(1-ethyl-1H-pyrazole-5-carbonyl)-3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{5-[1-(2-chlorobenzoyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
1-({1-[(3,4-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1,4-diazepan-5-one
3-(4-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperazin-1-yl)phenol
2-[2-(4-chlorophenyl)morpholin-4-yl]-N-(pyridin-2-ylmethyl)acetamide
2-[2-(1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
(1S,5R)-6-(furan-3-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-3-(1H-pyrazol-1-yl)benzamide
N-(1-benzylpiperidin-3-yl)-5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl})amine
1-(cyclohexylmethyl)-N-methyl-6-oxo-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
2-{4-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{[1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]methoxy}acetic acid
methyl 7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-3-(quinolin-8-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-(5-amino-1,3,4-thiadiazol-2-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
7-chloro-1-(pyridin-2-ylmethyl)-3-{[(thiophen-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
(4aR,7aS)-1-[(2-ethylphenyl)methyl]-4-(furan-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 4-(4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-cyclobutyl-N-{[(2S)-1-ethylpyrrolidin-2-yl]methyl}-6-methylpyrimidin-2-amine
1-(2,2-dimethylpropyl)-3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-(4-acetylbenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
6-methyl-2-[(2-methylphenyl)methyl]-1-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-1,4-dihydropyridin-4-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}-1,3-oxazole-4-carboxamide
(1S,5R)-3-(8-chloro-2-methylquinoline-4-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(3-{[1-(cyclohex-1-en-1-yl)ethyl]amino}propanamido)benzamide
methyl N-{1-oxo-1-[3-oxo-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]propan-2-yl}carbamate
1-[4-(3-methylphenoxy)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
1-(4-{[4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}piperidin-1-yl)ethan-1-one
3-(3,4-difluorophenyl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N,N-dimethyl-2-({[4-(methylsulfanyl)phenyl]formamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
(4S)-N-(3,4-difluorophenyl)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carboxamide
6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
4-(2,6-dimethylpyridin-3-yl)-N-[2-(propan-2-yloxy)ethyl]pyrimidin-2-amine
4-chloro-N,N-dimethyl-5-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-1,3-thiazol-2-amine
N-[4-(azepan-1-yl)butyl]-3-hydroxy-2-methylbenzamide
3-[(4-fluorophenyl)formamido]-N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]propanamide
(3R,4S)-1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-4-phenylpyrrolidin-3-amine
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-3-phenylpiperidine
3-(1H-1,3-benzodiazol-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]propanamide
N-[2-(azepan-1-yl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide