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4-{[3-(trifluoromethoxy)phenyl]methyl}-4H-1,2,4-triazole
4-({2-[1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2R,6R)-4-[(2-methoxyphenyl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-2-methyl-5-[5-(trifluoromethyl)-1,2-oxazol-3-yl]thiophene-3-sulfonamide
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}urea
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
3-{[(5-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}furan-2-yl)methyl]sulfanyl}-4H-1,2,4-triazole
3-[2-(5-ethylfuran-2-yl)-1H-imidazol-1-yl]-2-methoxypyridine
1-(1-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-phenylpiperidin-4-yl)ethan-1-one
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-indole
N-(2-hydroxyethyl)-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]-N-propylacetamide
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-{1-[1-(carbamoylmethyl)piperidin-4-yl]-N-[(2-methoxyphenyl)methyl]formamido}acetic acid
1-[2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]-1,4-diazepan-5-one
(4aS,8aR)-6-{3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carbonyl}-1-(3-methylbutyl)-decahydro-1,6-naphthyridin-2-one
{2-[2-amino-4-(cyclobutylamino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-oxoethyl}urea
3-(2-amino-1,3-thiazol-4-yl)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(thian-4-yl)piperazin-2-yl}ethan-1-ol
5-[2-(ethylamino)ethyl]-1-[(5-fluoro-2-methylphenyl)methyl]pyrrolidin-2-one
7-(2-methoxypyridine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-(dimethylamino)-3-(4-methoxy-2-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
methyl 3-benzamido-6-{[cyclohexyl(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
N,2,5-trimethyl-N-[(5-methylthiophen-2-yl)methyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-2-ylmethyl)piperidin-3-yl]-N-[4-(methylsulfanyl)phenyl]propanamide
1,3-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-[({5-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
3-(3-methylbutyl)-8-(oxan-3-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(prop-2-en-1-yl)-9-(1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[4-(pyrimidin-2-yloxy)phenyl]methyl})amine
4,5-dimethyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-[(5-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
(2S,3R)-2-amino-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-methoxybutanamide
3-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-4H-chromen-4-one
4-[1-(1-propylpiperidin-4-yl)piperidine-4-carbonyl]morpholine
N,N-dimethyl-5-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
{5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-yl]-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}(phenyl)methanol
N4-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5-ethylpyrimidine-2,4-diamine
4-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)-N-methylbenzene-1-sulfonamide
2-amino-4-(2-fluoro-4,5-dimethoxyphenyl)-6-(1-methyl-1H-pyrrol-3-yl)pyridine-3-carbonitrile
methyl 4-{4-[3-(pyridin-4-yl)propanoyl]piperazin-1-yl}benzoate
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amine
5-fluoro-N-(oxolan-2-ylmethyl)-4-(pyrrolidin-1-yl)pyrimidin-2-amine
4-[1-(1-benzyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]pyridine
(3aR,6aR)-2-(cyclobutylmethyl)-5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-methoxyphenyl)-1-{4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}propan-1-one
6-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one