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1-(3-fluoro-5-methylphenyl)-3-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
N,N-diethyl-1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidine-4-carboxamide
1-(5-chloropyridin-2-yl)-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazine
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
methyl 3-{3-[(3,4-dimethylphenyl)amino]piperidine-1-carbonyl}benzoate
{[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}(methyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
N-cyclopentyl-N'-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]butanediamide
4-(1-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}ethyl)morpholine
3-methyl-N-[(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)methyl]furan-2-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[(3S)-3-ethylmorpholin-4-yl]propan-1-one
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]propanamide
2-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]benzene-1,3-diol
2-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}pyridine
{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(furan-2-ylmethyl)(prop-2-yn-1-yl)amine
N-(2,2-difluoroethyl)-8-oxo-7-(prop-2-en-1-yl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
9-(1-benzofuran-5-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(4-hydroxyphenyl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-(furan-2-carbonyl)-4-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepane
2-oxo-N-phenyl-2-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2-fluoroethyl)piperidine-3-carboxamide
{2,4,6-trimethyl-3-[({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]phenyl}methanol
2-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxane-4-carboxamide
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-1H-pyrazole-3-carboxamide
N,N-dimethyl-7-(4-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[(4-methoxyphenyl)methyl]-N-[1-(pyridin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
5-methanesulfonyl-2-phenyl-4-(piperidin-3-yl)pyrimidine
6-[2-(pyridin-3-yl)-1H-imidazol-1-yl]-3,4-dihydroquinazolin-4-one
2-amino-4-{3-[2-(dimethylamino)ethoxy]phenyl}-6-(furan-2-yl)pyridine-3-carbonitrile
9-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-2-(methylsulfanyl)ethan-1-one
(4aR,7aS)-1-cyclobutanecarbonyl-4-[(4-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(2,6-dimethoxypyridin-3-yl)-3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
3-methyl-4-(2-phenyl-1,3-thiazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-ethyl-5-methyl-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,2-oxazole
[(3R,4R)-1-(1,5-dimethyl-1H-pyrrole-2-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
(3R)-2-(5-chloro-4-oxo-3,4-dihydroquinazolin-3-yl)-3-hydroxybutanamide
1-{[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}-2,2-bis(prop-2-en-1-yl)piperidine
methyl (1R,3S,3aR,6aS)-1-benzyl-5-methyl-4,6-dioxo-3-(pyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)ethan-1-one
3-[5-(2,5-dimethoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-3-yl]pyridine
1-[(3,4-difluorophenyl)methyl]-3-{1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl}-3-hydroxypiperidin-2-one
1-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
1-[7-(1,3-benzothiazol-2-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(dimethyl-1,2-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-[cyclohexyl(methyl)amino]-3-[3-({[2-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]propan-2-ol