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3-[3-({[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
2-(2,5-dimethoxyphenyl)-N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}acetamide
2-methyl-6-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-3-yl]pyrimidin-4-ol
methyl 5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
5-({4-[3-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methyl)-1H-1,2,3,4-tetrazole
N-{[3-(dimethylamino)phenyl]methyl}-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
1-(3,4-dimethoxybenzoyl)-3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine
2-methyl-N-({3-methyl-7-[3-(thiophen-2-yl)propanoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-4-carboxamide
1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-3-{2-oxo-2-[4-(pyridin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(1-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)piperidine-4-carboxylic acid
N-[(3R,4R)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-3-carboxamide
1-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-3-(4-hydroxyphenyl)propan-1-one
1-methyl-4-(2-{[methyl(prop-2-en-1-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)-1,2-dihydroquinolin-2-one
2-[2-(4-aminoazepan-1-yl)-2-oxoethyl]-4-phenyl-1,2-dihydrophthalazin-1-one
N-(furan-3-ylmethyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-1-methyl-1H-pyrazole-5-carboxamide
4-{[(2,2-dimethyloxan-4-yl)(ethyl)amino]methyl}-N-(pyridin-3-yl)benzamide
1-cyclohexyl-5-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-{1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidin-3-yl}benzoic acid
4-benzyl-1-[2-(4-ethylpiperazin-1-yl)-2-oxoethyl]-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-(pyridin-3-ylmethyl)urea
N-[4-(4-{[2-(2-chlorophenyl)ethyl]amino}piperidin-1-yl)phenyl]-2-(4-methoxyphenyl)acetamide
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(1-methyl-1H-indol-3-yl)ethan-1-one
[(2S,6S)-4-[2-(trifluoromethyl)benzoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
(1S,4S)-5-(cyclohexylmethyl)-2-(2-fluorophenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1λ6-thiomorpholine-1,1-dione
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-{[(furan-2-ylmethyl)(methyl)amino]methyl}-3-hydroxypiperidin-2-one
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-{[5-(4-chlorophenyl)furan-2-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
methyl 2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]amino}acetate
2-{[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]methyl}benzoic acid
5-chloro-2-methoxy-4-[5-(piperidin-1-ylmethyl)pyridin-2-yl]pyridine
2-(2,4-dimethylbenzenesulfonamido)-N-[2-(ethylsulfanyl)ethyl]acetamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylpyridine-3-carboxamide
1-cyclopentanecarbonyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(2-{7-[(2,6-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
5-{2-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-benzyl-5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-ethoxy-4-[4-phenyl-1-(pyridin-3-ylmethyl)-1H-imidazol-5-yl]phenol
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-4-sulfamoylpiperazine-1-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1-phenylpiperidin-4-yl)acetamide
(1S,5R)-3-[2-(2-hydroxyethoxy)ethyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-2-fluoro-N-[(7-methoxy-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}quinolin-3-yl)methyl]benzamide
1-(2-methoxyphenyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
1-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-(1,2-oxazinan-2-yl)propan-1-one
[(3S,5R)-1-(3-chloro-4-ethoxybenzoyl)-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
3-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
1-[2-(2,3-dimethylphenoxy)ethyl]-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine