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5-(1,2-oxazinane-2-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrazine
3-{2-[(3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]propanamide
1-(4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
4-(2-methoxyacetyl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]ethan-1-one
(1S,5R)-3-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(azepane-1-carbonyl)-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-(2-methylpropyl)-1,4-dihydropyridin-4-one
(2S,4R)-N,N-diethyl-4-(2-hydroxyacetamido)-1-(5-methylpyrazine-2-carbonyl)pyrrolidine-2-carboxamide
8-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-{1-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}benzoic acid
methyl 8-[1-(ethoxycarbonyl)piperidin-4-yl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
methyl 3-(2-chloro-4-fluorobenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{4-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]-1,4-oxazepan-6-yl}methanol
1-{4-[(1S,4S)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(1S,5R)-3-(5-chloro-3-fluoropyridin-2-yl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4-methylphenyl)methyl]-4-(4-methylpiperidine-4-carbonyl)piperazin-2-one
2-{2-[(1H-indol-6-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
1-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-(4-methyl-1H-pyrazol-3-yl)piperidine
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-(oxan-4-yl)piperidine-4-carboxamide
6-[4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-N-propylpyridine-3-carboxamide
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}ethan-1-one
1-(2-chlorophenyl)-4-(4-propyl-1,2,3-thiadiazole-5-carbonyl)piperazin-2-one
3-({6-[(dimethylamino)methyl]-1,4-oxazepan-4-yl}methyl)-8-methylquinolin-2-ol
2-(1H-1,3-benzodiazol-1-yl)-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
N-(cyclopropylmethyl)-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(oxolan-2-ylmethyl)benzamide
N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1H-indazole-3-carboxamide
3-{1-[(1R,9aR)-octahydro-1H-quinolizine-1-carbonyl]piperidin-4-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(3-chloro-4-fluorophenyl)-3-[1-(3-methoxypropanoyl)piperidin-4-yl]propanamide
N4-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5,6-dimethylpyrimidine-2,4-diamine
methyl[(2-methyl-1,3-oxazol-4-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,3-thiazole-5-carboxamide
4-[1-(pyrimidin-5-yl)-1H-pyrazol-3-yl]benzoic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
methyl 3-(2,3-dimethylbenzoyl)-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(4aS,8aR)-1-(2-aminoethyl)-6-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
N4-methyl-N6-(propan-2-yl)-N4-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-4,6-diamine
4-ethyl-3-({1-[(4-fluorophenyl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-1-(propan-2-yl)piperidine-4-carboxamide
(4aR,7aS)-4-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}butanamide
4-methyl-N-(2-phenylethyl)-2-(propan-2-yl)-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
3-(benzyloxy)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(1H-pyrazole-3-carbonyl)piperidine
4-{5-methyl-2-oxo-4-[4-(propan-2-yloxy)benzoyl]piperazin-1-yl}benzonitrile
N-{1-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
1-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
1-(pyridin-2-ylmethyl)-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide