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N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylcyclopropanecarboxamide
1-[(3-fluorophenyl)methyl]-5-[4-(2-methoxyethoxy)piperidine-1-carbonyl]piperidin-2-one
4-{4-[(2,3-dimethoxyphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[1-(2,6-dimethylphenoxy)propan-2-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-[(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)oxy]pyridine
7-(5-chloropyridin-2-yl)-4-cyclopentanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-(2-chlorophenyl)-7-methyl-N-(oxan-4-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[2-(diethylamino)ethyl]-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-(4-methylphenyl)-4-[(2S)-5-oxopyrrolidine-2-carbonyl]piperazin-2-one
N-(4-{[(3aS,6aS)-1-(2-phenylethyl)-octahydropyrrolo[2,3-c]pyrrol-5-yl]methyl}phenyl)acetamide
3-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}benzonitrile
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-N-(3-fluorophenyl)-2-oxoacetamide
2-[(3S,4R)-3-propyl-4-(1,3-thiazole-4-amido)pyrrolidin-1-yl]acetic acid
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine
8-[(5-propylfuran-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]thiomorpholine
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-benzothiophene-5-carbonyl)piperazine
5-(1H-imidazol-2-yl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]thiophene-2-carboxamide
2-{4-[(2,6-difluorophenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
[3-(3-methylbut-2-en-1-yl)-1-(1,3-thiazol-4-ylmethyl)piperidin-3-yl]methanol
N-ethyl-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(2-methyl-5-oxopyrrolidin-1-yl)acetamide
4-[({[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}amino)methyl]benzene-1-sulfonamide
1-[(4aR,8aR)-1-(cyclohex-1-ene-1-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(2-methoxyphenyl)ethan-1-one
N-(4-fluorophenyl)-1-[2-(1H-indol-3-yl)acetyl]piperazine-2-carboxamide
2-(3-acetyl-1H-indol-1-yl)-1-{2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}butan-1-one
N-(2-methoxyethyl)-1-[(1s,4s)-4-aminocyclohexyl]-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]acetamide
2-amino-4-[2-(prop-2-en-1-yloxy)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-[(2-methylphenyl)sulfanyl]piperidine
N,N-dimethyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
4-(2,3-dimethylphenyl)-6-methylpyrimidin-2-amine
N-ethyl-3-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}benzamide
3-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]sulfonyl}-N-(prop-2-en-1-yl)benzamide
N,6-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
1-methyl-5-({2-[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3,4-tetrazole
(4aR,7aS)-1-cyclopropanecarbonyl-4-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
5-propyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-{[3-(2-methyl-1,3-thiazol-4-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-(cyclobutylsulfamoyl)-N-[2-(ethylsulfanyl)ethyl]benzamide
3-{4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,2,3-triazol-1-yl}propane-1,2-diol
7-fluoro-2-methyl-4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]quinoline
N-[1-(4-acetyl-4-phenylpiperidin-1-yl)-1-oxopropan-2-yl]methanesulfonamide