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N-{5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl}-2-methylbutanamide
4-(4-ethoxyphenyl)-3-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-2-(4-methylphenyl)pyrimidin-4-ol
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}[(6-methylpyridin-2-yl)methyl]amine
1-(1-benzothiophene-5-carbonyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
N,2-dimethyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
8-[(3,5-difluorophenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-2-(pyrrolidin-1-yl)pyridine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
2-ethyl-8-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)pyridine
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1-oxaspiro[4.4]nonan-2-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-(hydroxymethyl)piperidin-3-ol
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-2-[(1-methyl-1H-indol-3-yl)sulfanyl]acetamide
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1-(2,4,5-trimethoxyphenyl)propan-1-one
[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl](benzylsulfamoyl)amine
9-[2-(3-fluorophenyl)ethyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperazine
[3-(dimethyl-1,2-oxazol-4-yl)propyl](6-methylhept-5-en-2-yl)amine
5-fluoro-3-methyl-2-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-indole
1-[(3-methoxyphenyl)methyl]-4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-2-one
4-(cyclopentylsulfamoyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
N-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-yl)methanesulfonamide
N-cyclopropyl-2-[2-(methylcarbamoyl)phenyl]pyridine-3-carboxamide
2-benzyl-4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]morpholine
3-(2,4-difluorophenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]quinoxaline-5-carboxamide
N-{1-[1-(1-methoxypropan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
N-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)methyl]-3-methylfuran-2-carboxamide
5-chloro-3-methyl-2-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-1H-indole
1-ethyl-8-(9H-fluoren-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}propanamide
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-cyclohexyl-N-methylpiperidine-3-carboxamide
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3-[(2-fluorophenyl)formamido]propanamide
4-(4-methoxyphenyl)-N-[2-(methylsulfanyl)phenyl]piperazine-1-carboxamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(thiophen-2-yl)ethan-1-one
2-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxo-S-(thiophen-2-yl)ethane-1-sulfonamido
N-[(3S,4R)-1-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]benzamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}propan-1-one
N-(2-methoxyethyl)-3-{[1-(pyrazine-2-carbonyl)piperidin-4-yl]oxy}benzamide
3-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-9-methyl-9H-carbazole
1'-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-oxo-1-phenyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-3-carboxamide
N-cyclopropyl-4-methoxy-3-({1-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-yl}oxy)benzamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
2-methyl-2-{2-[(1-methylpiperidin-3-yl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid