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(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[5-(propan-2-yl)thiophene-3-carbonyl]piperidin-4-ol
1-[(3,4-dimethylphenyl)methyl]-4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(1S,4S)-5-[(5-chloro-2-hydroxyphenyl)methyl]-2-[2-(methylsulfanyl)phenyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
ethyl 1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(oxolan-3-yl)propanamide
[(2S,6S)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
3-phenyl-5-(2-propoxybenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{3-[2-(methylsulfanyl)ethyl]-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-(3,4-dimethoxyphenyl)-1-(3-methoxybenzoyl)piperidin-3-amine
N,N-dimethyl-3-{[3-(pyrimidin-4-yl)piperidin-1-yl]sulfonyl}benzamide
N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]cyclobutanecarboxamide
4-[(3,4-difluorophenyl)methyl]-3-[2-(2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]piperazin-2-one
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N,N-diethylpropanamide
2-{5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-3-yl}acetamide
N-(1-{[(2,2-diphenylethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-2-carboxamide
4,6-dimethyl-1-(2-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
7-[(2-fluorophenyl)methyl]-2-(4,4,4-trifluorobutyl)-2,7-diazaspiro[4.5]decane
N-[2-(4-phenylpyrimidin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
5-(4-ethylpiperazine-1-carbonyl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole
3-methyl-4-(1-{5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}pyrrolidin-2-yl)-1,2,5-oxadiazole
2-(2-cyclopropyl-1H-1,3-benzodiazol-1-yl)-N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]acetamide
(2S,4S)-4-amino-N-{[1-(2-hydroxyethyl)piperidin-4-yl]methyl}-N,1-dimethylpyrrolidine-2-carboxamide
4-(4-cycloheptylpiperazin-1-yl)-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-chloro-N-(4-{4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidin-1-yl}phenyl)benzamide
[(3R,4R)-1-(3,4-dimethylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-acetyl-8-[(5-cyano-1-methyl-1H-pyrrol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
{1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
2-(1,3-dimethyl-4-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]propanamide
5-(4-benzylpiperidin-1-yl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
6-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]quinoxaline
3-{5-[2-amino-6-(propan-2-yl)pyrimidine-4-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
N-[(6-hydroxypyrimidin-4-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
8-fluoro-N-[3-(pyridin-3-yloxy)propyl]quinoline-2-carboxamide
1-[benzyl(methyl)amino]-3-{4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propan-2-ol
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinoxalin-2-yl)piperidin-3-yl]propanoic acid
8-{[2-(carboxymethoxy)-5-chlorophenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2,6,8-trimethyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2-(trifluoromethyl)benzamide
7-[(2,3-difluorophenyl)methyl]-2-(5-methoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
methyl 3-(furan-3-amido)-5-[(4-methylpentan-2-yl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[4-(1-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)phenyl]acetamide
3-[(1-{5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)oxy]pyridine
N,1-dimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-acetyl-N-{[4-fluoro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
2-(1-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-3-oxopiperazin-2-yl)-N-methylacetamide
N-(2,4-difluorophenyl)-4-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)benzamide
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-N-(3-fluorophenyl)piperidin-3-amine
3-[2-(2-methylphenyl)ethyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine