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({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(2-methoxyethyl)methylamine
1-(cyclopropylmethyl)-6-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(3-methoxyphenyl)-4-[(1R,2R)-2-phenylcyclopropanecarbonyl]piperazin-2-one
7-(2-methoxyethyl)-2-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2,7-diazaspiro[4.5]decan-6-one
3-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-2-yl)pyridine
3-(4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1λ6-thiolane-1,1-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}benzamide
1-[1-(1-ethylpiperidine-4-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-butyl-2-methanesulfonyl-N-(thiophen-3-ylmethyl)acetamide
4-hydroxy-N-[3-(pyridin-3-yloxy)propyl]-2-(thiophen-2-yl)pyrimidine-5-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-5-phenyl-1,2,4-triazin-3-amine
(1S,4S)-2-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-2-azabicyclo[2.2.1]heptane
4-[3-(morpholin-4-yl)piperidin-1-yl]-2-phenylquinazoline
[(3R,4R)-1-{[5-(2-fluorophenyl)furan-2-yl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2,7,8-trimethylquinoline-4-carboxamide
3-{3-methyl-5-[2-(2-oxoazepan-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
4-(dimethyl-1,2-oxazole-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N-[(7-{[5-(4-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-(3-fluorophenyl)acetamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[2-(4-methylphenyl)ethyl]piperidine-4-carboxamide
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine
2-[(3,4-difluorophenyl)methyl]-8-(furan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
1-methyl-4-(1-propylpiperidin-4-yl)-1,4-diazepane
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(2H-1,3-benzodioxol-5-yl)-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
2,5-dimethyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(1R,2S,4R)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
{3-[(4-fluorophenyl)methyl]-1-(quinoline-6-carbonyl)piperidin-3-yl}methanol
1-{4-[2-(3-methoxyphenyl)azetidine-1-carbonyl]phenyl}-1H-imidazole
3-(2-hydroxyphenyl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1H-pyrazole-5-carboxamide
1-{2-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]ethyl}pyrrolidin-2-one
1-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(4aS,8aS)-2-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-decahydroisoquinolin-4a-ol
5-methyl-3-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-2H-indazole
(3aS,6aS)-2-(dimethylcarbamoyl)-5-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
{[2-(azocan-1-yl)pyridin-3-yl]methyl}[(1-ethyl-1H-pyrazol-4-yl)methyl]amine
2-(4-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-7-fluoroquinolin-2-yl}-1H-pyrazol-1-yl)ethan-1-ol
2-{4-[(4-hydroxy-6-methylquinolin-2-yl)methyl]piperazin-1-yl}-1-(pyrrolidin-1-yl)ethan-1-one
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[(3R,4R)-3-hydroxy-1-[1-(propan-2-yl)-1H-pyrrole-2-carbonyl]piperidin-4-yl]pyridine-2-carboxamide
methyl 2-{3-oxo-4-[2-(4H-1,2,4-triazol-4-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
N-[(1R,3R)-3-aminocyclopentyl]-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
5-({4-oxo-3H,4H-pyrido[2,3-d]pyrimidin-3-yl}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-methyl-2-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
4-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}pyridine
1-(cyclopropylmethyl)-5-(quinoxaline-5-carbonyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,2,3,4-tetrahydronaphthalene-2-carboxamide
methyl 1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
1-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazin-1-yl)-4-phenylbutane-1,4-dione