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N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-[(2-phenylquinolin-4-yl)formamido]acetic acid
5-oxo-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
3-(2-ethoxypropyl)-3-methyl-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
N,N-dimethyl-2-{[4-methyl-4-(methylsulfanyl)pentan-2-yl]amino}ethane-1-sulfonamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
2-{4-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(2,5-dimethylfuran-3-yl)-3,4-dihydropyrimidin-4-one
N-{2-[1-(hydroxymethyl)-9-[(2-methylphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl}acetamide
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(9H-fluoren-2-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-1-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-methyl-8-[(3-methylquinoxalin-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
(1R,5S,6R)-3-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-cyclopentyl-6-oxopiperidine-3-carboxamide
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-methyl-5-(1H-1,2,3-triazol-5-yl)-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
[5-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}methyl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methylphenol
2-[(4aS,8aR)-1-(3-aminopropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-6-methylpyridine-3-carboxamide
6-{[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
ethyl 5-[(4-hydroxyphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(2S)-N-ethyl-1-[4-hydroxy-2-(4-methylphenyl)pyrimidine-5-carbonyl]pyrrolidine-2-carboxamide
2-[2-(dimethylamino)ethyl]-8-(7-fluoro-4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1,4,6-trimethyl-N-[(4-methyl-2-phenyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-(2-methoxyphenyl)-3-{1-[1-(thiolan-3-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3-methylthiophen-2-yl)methyl]({[2-(propan-2-yl)pyrimidin-4-yl]methyl})(pyridin-2-ylmethyl)amine
N-[2-(5-cyano-2-methyl-1H-indol-3-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
{4-[(3-methoxyphenyl)methyl]-1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-4-yl}methanol
3-(cyclopropylsulfamoyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
2-fluoro-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-6-methoxybenzamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidine-3-carboxylate
2-[methyl(2-methylpropyl)amino]-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-dimethylpiperazine-1-carboxamide
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(2-hydroxyethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
7-[(4-fluorophenyl)methyl]-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
1-(pyrimidin-2-yl)-4-[6-(1,2,3,6-tetrahydropyridin-1-yl)pyridine-3-carbonyl]-1,4-diazepane
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}butanoic acid
ethyl 3-[(2-fluorophenyl)methyl]-1-(4-methoxy-4-oxobutanoyl)piperidine-3-carboxylate
3-(2-fluorophenyl)-N-methyl-N-(1,2-oxazol-3-ylmethyl)-3-phenylpropanamide
(2S,4R)-4-{[(2,5-dimethylphenyl)methyl]amino}-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-methyl-2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,2-dihydrophthalazin-1-one
7-(2-methylphenyl)-4-(1H-1,2,4-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-(oxane-4-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1,2-oxazol-3-ylmethyl)-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
3-(5-methylfuran-2-yl)-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1H-pyrazole-5-carboxamide