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5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-1,3-benzodiazole-7-carboxamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[4-(trifluoromethyl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
2-(oxolan-2-ylmethyl)-9-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-3-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-[2-(pyrrolidin-1-yl)ethyl]propanamide
6-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylpyrimidin-4-amine
methyl 5-{[(4-chlorophenyl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[2-(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
dimethyl[(4-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
2-ethyl-1-[4-(3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}phenoxy)piperidin-1-yl]butan-1-one
N-cyclopropyl-1-[1-(2-methylbenzoyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
1-ethyl-5-{[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N-[3-(2-methoxyacetamido)phenyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine-1-carboxamide
4-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-(furan-2-ylmethyl)piperidine
5-[1-(4-chlorophenyl)cyclopropanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
5-[(methylsulfanyl)methyl]-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]furan-2-carboxamide
(4-{[3-(benzyloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)(pyridin-3-yl)methanol
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(oxolan-3-yl)amino]pyridine-3-carboxamide
(3R,4S)-4-(4-methoxyphenyl)-1-(5-phenyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-amine
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-methoxy-3-(methoxymethyl)phenyl]methyl})amine
3-(3-fluoro-4-methoxybenzoyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-1-methyl-5-phenyl-1H-pyrrole-2-carboxamide
1-(2-{4-[(2-methoxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
5-(2-hydroxypropanoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[4-(2-aminopyrimidin-4-yl)piperidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
1-[(2-methoxyphenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-cyclopropyl-1-{6-hydroxy-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl)[2-(morpholin-4-yl)propyl]amine
(3S,4R)-3-ethyl-1-[3-(hydroxymethyl)-7-methylquinolin-2-yl]-4-methylpiperidin-4-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
2-methyl-9-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-phenyl-2,9-diazaspiro[5.5]undecane
5-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-{2-[7-(2-ethylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-4-methoxybenzamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
4-(3-chloropyridin-2-yl)piperazine-2-carboxylic acid
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4S)-4-({[4-(benzyloxy)-2-methoxyphenyl]methyl}(ethyl)amino)oxolan-3-ol
(3aS,6aS)-2-methyl-5-[2-(6-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-[(2,6-difluorophenyl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]benzamide
1-(3,3-diphenylpiperidin-1-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-(4-fluorobenzenesulfonyl)ethyl]acetamide
N-[(4-methylphenyl)methyl]-3-{4-[(1-methylpiperidin-4-yl)methyl]piperazin-1-yl}propanamide
3-(dimethylamino)-N-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propyl]benzamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
1-({3-[hydroxy(phenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}methyl)azepan-2-one
N-{1-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide