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6-[(3-fluorophenyl)methyl]-2-[3-(piperidin-1-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
[(1S,3S,3aS,6aR)-5-methyl-3-(naphthalen-1-yl)-1-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
6-cyclopropyl-N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}pyrimidin-4-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-methylprop-2-en-1-yl)piperazine
2-(2,6-dimethoxyphenyl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
2-methyl-5-phenyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[2-(morpholin-2-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
1-(cyclobutylmethyl)-3-{[4-(cyclobutylmethyl)piperazin-1-yl]methyl}-3-hydroxypiperidin-2-one
(2S)-2-{[1-(4-chlorophenyl)propan-2-yl]amino}-3,3-dimethylbutan-1-ol
4-methyl-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}pyrimidin-2-amine
1-ethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
2-(pyridin-3-yl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
1-{4-[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]thiophen-2-yl}ethan-1-one
3-methyl-7-[8-(trifluoromethyl)quinolin-4-yl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-methyl-3-[({2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}carbamoyl)amino]benzamide
5-[(4-fluorophenyl)methyl]-5-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)imidazolidine-2,4-dione
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
N-(1-methoxybutan-2-yl)-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
1-methyl-4-(3,4,5-trimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridine
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
(4S)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3,3,4-trimethylpiperidin-4-ol
(1R,2R)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-phenylcyclopropane-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-(2-carbamoylethyl)-3-phenylpropanamide
2-(azepan-1-yl)-2-(3,4-dimethoxyphenyl)acetic acid
1-(6-fluoro-4-methylquinazolin-2-yl)-N-(1H-indol-4-ylmethyl)piperidin-4-amine
N3-[(2-chloro-4-fluorophenyl)methyl]piperidine-1,3-dicarboxamide
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-3-methylfuran-2-carboxamide
(2S,4S)-N-ethyl-4-(furan-3-amido)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
2-cyclopropyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
9-[(4-chloro-2-fluorophenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(2-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methyl]propanamide
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
6-{2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
2-[ethyl(methyl)amino]-2-[6-(piperidin-1-yl)pyridin-3-yl]acetic acid
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
2-cyclobutyl-5-(2-methoxyacetamido)-N,1-dimethyl-N-(quinoxalin-6-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
4,5-dimethyl 1-[(3S,5S)-5-[(furan-2-ylmethyl)carbamoyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
(3R,4S)-4-cyclopropyl-1-(3-methoxybenzenesulfonyl)pyrrolidin-3-amine
1-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(2-methoxyphenoxy)ethan-1-one
(3S,4S)-N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-hydroxy-4-(4-methylpiperazin-1-yl)pyrrolidine-1-carboxamide
N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
methyl 3-{7-chloro-2-[(oxan-4-ylformamido)methyl]-2,3-dihydro-1-benzofuran-5-yl}benzoate
N-[(2R,3R)-2-methoxy-1'-[2-(3-methoxyphenyl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
2-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-hydroxy-3-methylbutan-1-one
1-[2-(dimethylamino)-4-[methyl({[2-(methylamino)pyrimidin-5-yl]methyl})amino]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-{[2-(furan-3-yl)-1H-imidazol-1-yl]methyl}-3-methylpyridine