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4-[2-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
2-(2-methoxyethyl)-3-oxo-N-[(1S)-1-phenylethyl]-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{4-[(1-benzyl-1H-pyrazol-4-yl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
4-(4-chlorophenoxy)-1-[2-(2-methyl-1,3-thiazol-4-yl)ethyl]piperidine
5-(1-cyclohexanecarbonylpyrrolidin-2-yl)-3-(2-methoxyphenyl)-1,2,4-oxadiazole
4-[5-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[(3,3,4-trimethylpiperazin-1-yl)methyl]piperidin-2-one
5-{[4-(methylsulfanyl)phenyl]methyl}-5-{3-oxo-3-[4-(quinazolin-2-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
2-[ethyl(methyl)amino]-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
4-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidine-1-carbonyl}pyridine
N-[4-chloro-3-({[(3-hydroxypiperidin-3-yl)methyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
(4aR,7aS)-1-(furan-2-ylmethyl)-4-[2-(2-methylphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2R,3R)-2-methoxy-1'-[(2-methylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
3-{[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]sulfamoyl}-N-cyclopropylbenzamide
1-methyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-2-carboxamide
3-(2-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}ethyl)quinoxalin-2-ol
4-(4-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-2-oxopiperazin-1-yl)benzonitrile
2-methyl-3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6H,7H-pyrazolo[1,5-d][1,2,4]triazin-7-one
2-(azepan-1-yl)-1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]propanamide
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-methyl-1,3-thiazole-4-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(quinolin-6-ylmethyl)acetamide
2-[4-(hydroxymethyl)-4-(3-phenylpropyl)piperidin-1-yl]-6-methylpyridine-3-carboxamide
7-[(2,3-difluorophenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-(5-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)pyridine
N-({1-[(3-chloropyridin-4-yl)methyl]pyrrolidin-3-yl}methyl)-2-(furan-2-yl)-2-oxoacetamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-2-(morpholin-2-yl)acetamide
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
2-(2,4-dichlorophenoxy)-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]acetamide
5-(propan-2-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-(3-ethoxypropyl)-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methanol
(2R,3R,6R)-5-(furan-2-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-chloro-N-{2-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]propyl}benzamide
N-[1-(4-chlorophenyl)cyclobutyl]-1-(2-methoxyethyl)piperidine-3-carboxamide
N-[(3S,4R)-1-[3-(1H-indol-3-yl)propanoyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,3,5-trimethyl-1H-indole-2-carboxamide
2-amino-4-(thiophen-3-yl)-6-(2,3,4-trimethoxyphenyl)pyridine-3-carbonitrile
(2E)-N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidine
(1S)-1-[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]-2-(1H-imidazol-4-yl)ethan-1-amine
N-{[7-(5-methyl-1H-indole-2-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}oxolane-3-carboxamide
2-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-propylpyrimidine
4-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-N-methylbenzene-1-sulfonamide
3-{2-oxo-2-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
4-methyl-6-[4-(5-methyl-1-benzofuran-2-carbonyl)piperazin-1-yl]pyrimidin-2-amine
1-cyclohexyl-N-cyclopropyl-5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
2-(2-propyl-1,3-thiazole-4-carbonyl)-2,3-dihydro-1H-isoindole
5-(oxolan-2-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}thiophene-2-carboxamide
1-(adamantan-1-yl)-4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazine