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1-[2-({[2-(2-methylphenyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-cyclobutyl-2-fluoro-5-sulfamoylbenzamide
(3S,4S)-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]-4-propylpyrrolidine-3-carboxylic acid
2-(3-methyl-1H-pyrazol-1-yl)-1-[4-(4-phenyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]ethan-1-one
1-[(3S,4R)-1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
N-(cyclopropylmethyl)-4-[methyl(pyridin-3-ylmethyl)sulfamoyl]benzamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-4-(pyrimidin-2-yl)piperazine-2-carboxylic acid
2-[4-(1H-indol-5-ylmethyl)morpholin-3-yl]acetic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-6-oxo-1,6-dihydropyridazine-3-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]acetamide
2-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1-benzofuran-5-carboxamide
N-cyclopropyl-3-({1-oxaspiro[4.5]decan-3-yl}sulfamoyl)benzamide
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-hydroxy-2,2-dimethylpropyl)propanamide
4-methyl-2-{1-[4-phenyl-5-(pyridin-3-yl)-1H-imidazol-1-yl]propyl}pyridine
1-[(2-methyloxolan-2-yl)methyl]-4-(3-methylthiophen-2-yl)-1H-1,2,3-triazole
2-[(4aR,7aS)-4-cyclopentanecarbonyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1H-indazole-3-carboxamide
4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-1,2-dimethylpiperazine
{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[3-(oxolan-2-yl)propyl]amine
(1S,5R)-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
2-methoxy-5-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)benzoic acid
ethyl 1-[(5-acetylthiophen-3-yl)methyl]-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
1-ethyl-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}piperidine-3-carboxamide
(3S,4R)-1-(3-fluoropyridine-4-carbonyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(thian-4-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(3-phenylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(5-oxopyrrolidin-2-yl)acetamide
3-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl}-1-(morpholin-4-yl)propan-1-one
(1S,5R)-6-(1-methyl-1H-indole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(2-methylpropyl)amine
N-(5-{[1-(2-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}thiophen-2-yl)acetamide
5-{1-[3-(diethylamino)propanoyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
N-(2-ethyl-6-methylphenyl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
N-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-oxo-8-(3-phenylpropyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
7-[(2,3-difluorophenyl)methyl]-2-methyl-2,7-diazaspiro[4.5]decane
[1-(3-fluoro-4-methoxybenzoyl)-3-(2-phenylethyl)piperidin-3-yl]methanol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanamide
2-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
5-(2,6-difluorophenoxymethyl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,2-oxazole-3-carboxamide
1-benzyl-4-[2-(morpholin-4-yl)ethyl]-1,4-diazepan-6-ol
5-cyclopropanecarbonyl-1'-(quinolin-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-(2-hydroxyphenoxy)acetamide
2-benzyl-5-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,3-benzoxazole
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine