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(4aS,7aR)-1-[2-(methylamino)acetyl]-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-({4-[3-(4-fluorophenyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
5-(2,6-difluorophenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[1-(4-fluorophenyl)ethyl]-1-methyl-1H-pyrazole-5-carboxamide
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl){[2-(methylsulfanyl)pyrimidin-5-yl]methyl}amine
1-{2-oxo-2-[3-oxo-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1'-(4-methyl-1,3-thiazole-5-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-phenylpiperazine
1-[(3R,4R)-3-hydroxy-4-(4-methylpiperazin-1-yl)piperidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
3-{[4-(3-chloro-5-fluoro-4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
(4R)-N-[(1-benzylpiperidin-4-yl)methyl]-N,3-dimethyl-1,3-thiazolidine-4-carboxamide
N-({8-[(4-ethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
4-[1-(3-chloro-2-fluorophenyl)-1H-imidazol-2-yl]-1-(2-methoxyethyl)piperidine
4-[(1-cyclopentylpiperidin-4-yl)oxy]-3-methoxy-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}[3-(dimethylamino)propyl][3-(1H-pyrazol-1-yl)propyl]amine
N-cyclopentyl-2-acetamido-3-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)butanamide
2-{[(3R,5S)-1-[(2-ethoxyphenyl)methyl]-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]sulfanyl}-1H-1,3-benzodiazole
(3aR,6aR)-2-[(5-chlorofuran-2-yl)methyl]-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-methoxyphenoxy)-N-{[1-(oxan-4-yl)piperidin-3-yl]methyl}acetamide
3-(2-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
5-[1-(2-methoxybenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-{1-[(2,4-difluorophenyl)methyl]piperidin-3-yl}-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
[4-fluoro-3-(2-phenylphenyl)phenyl]methanamine
4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-ethyl-N-methyl-2-oxo-N-(quinolin-5-ylmethyl)-1,2-dihydropyridine-4-carboxamide
9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-3-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
ethyl 1-[(1-methyl-1H-imidazol-2-yl)methyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
2-[4-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethan-1-amine
3-(1,3-difluoropropan-2-yl)-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
1-ethyl-5-[2-(2-fluorophenyl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
methyl 6-(2-fluorobenzoyl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-chloro-5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}pyridine
N-(1-methyl-1H-1,3-benzodiazol-5-yl)-4-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
N-benzyl-2-[(6-{[(4-fluorophenyl)methyl](methyl)amino}pyridazin-3-yl)oxy]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]acetamide
3-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-methyl-1-(quinolin-5-yl)urea
[4-methyl-5-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methanol
8-(1H-indol-2-ylmethyl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-{[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridazine
4-ethyl-3-({1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-methyl-1-(4-methyl-2-oxo-2H-chromen-7-yl)urea
methyl 3-[(3-fluoro-4-methoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3-{[(2-{imidazo[1,2-a]pyrimidin-2-yl}ethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
2-benzyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1,3-thiazole-4-carboxamide
N-[3-(4-{[(4-methoxyphenyl)formamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-methylthiophene-2-carboxamide
6-[3-(3-methoxypropyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione