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7-(1-methanesulfonylpyrrolidine-2-carbonyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl 2-[4-(2-phenylpyrimidin-4-yl)piperidine-1-carbonyl]benzoate
N-(3,4-dimethylphenyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-amine
1-(5-cyclopropyl-1,2-oxazole-3-carbonyl)-3-[3-(propan-2-yloxy)benzoyl]piperidine
(4aR,7aS)-1-(pyrimidin-2-yl)-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(5S,9aS,9bS)-5-(4-ethoxyphenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1-methanesulfonylpiperidin-4-yl)-5-propylthiophene-3-carboxamide
3-(pyridin-3-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]propan-1-one
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-oxopentanamide
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[3-(1,3-oxazol-5-yl)phenyl]piperidin-4-amine
3-(methoxymethyl)-1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
1-(2,2-dimethylpropyl)-4-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}pyrrolidin-2-one
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyloxane-2-carboxamide
2-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-7-methyl-4H-chromen-4-one
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-1H-1,2,3-triazole
N-benzyl-6-(2,5-dimethylphenyl)-N-(2-hydroxyethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(morpholin-3-yl)-N-[4-(3-phenyl-1,2,4-oxadiazol-5-yl)phenyl]acetamide
N-[(5-methylpyrazin-2-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
9-methoxy-3-[(4-methoxy-3-methylphenyl)methyl]-N-[(3-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1S,2S,9S)-N-(1H-indol-5-yl)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
4-{4-[3-(trifluoromethyl)phenoxy]piperidine-1-carbonyl}pyridin-2-amine
N-(2-hydroxyethyl)-5-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-methyl-N-{1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
N5-{imidazo[1,2-a]pyridin-3-ylmethyl}-N5-methyl-N6-(thiophen-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
N-ethyl-1-[3-(prop-2-en-1-yloxy)benzoyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-(1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-1,3-benzothiazole
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-phenoxyfuran-2-carboxamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}acetamide
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2,6-dimethylquinoline-4-carboxamide
N-[2-(4-fluorophenyl)ethyl]oxane-2-carboxamide
6-(methylsulfanyl)-2-[3-(1H-pyrazol-1-yl)benzoyl]-1,2,3,4-tetrahydroisoquinoline
1-[4-(aminomethyl)phenyl]-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)urea
(9aS)-N-{4-[2-(pyridin-2-yl)ethyl]phenyl}-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)-N-[(3S)-2-oxoazepan-3-yl]benzamide
N,N-dimethyl-2-{8-[(5-methylpyrazin-2-yl)methyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}acetamide
2-(2,6-difluorophenyl)-N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-ethyl-3-{[2-(2-fluorophenyl)-2-hydroxyethyl]sulfamoyl}-N-methylbenzamide
N,N-bis(1,3-oxazol-4-ylmethyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-{[ethyl(2-methoxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-[(3R,4S)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
N,N-diethyl-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-sulfonamide
1-[benzyl(methyl)amino]-3-[2-methoxy-5-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
N-[(2-fluorophenyl)methyl]-2-[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]acetamide
3-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea
(5S,9aS,9bS)-2-methyl-5-(5-methylthiophen-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(methylamino)pyrimidine-5-carboxamide
4-[(1R,7S)-3-(2,2-dimethylpropyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]piperazine-1-carboxamide
N-cyclopropyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-(pyridin-3-ylmethyl)acetamide
N-[2-(5-methylfuran-2-yl)phenyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide