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[3-(3-methylbut-2-en-1-yl)-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methanol
1-{[5-(4-fluorophenyl)-2-hydroxyphenyl]methyl}piperidin-3-ol
ethyl 1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-carboxylate
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-(1,3-thiazole-5-carbonyl)-1,4-diazepan-2-one
3-[(3R,4S)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
(1S,5R)-3-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[4-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-1-methylpiperazin-2-yl]methanol
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-hydroxybenzamide
(3R,4S)-4-cyclopropyl-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-amine
3-(2-methylphenyl)-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
N,2,6-trimethyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]quinoline-4-carboxamide
ethyl 2-[1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperidin-2-yl]acetate
2-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(3-methoxyphenyl)-3-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]piperidin-4-yl}propanamide
1-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
5-[benzyl(methyl)amino]-2-[(2R)-3-hydroxy-2-methylpropyl]-2,3-dihydropyridazin-3-one
(5S)-5-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}pyrrolidin-2-one
(3S,4S)-4-cyclopropyl-1-[3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoyl]pyrrolidine-3-carboxylic acid
4-methyl-2-(1-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
methyl 1-[(3R,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(quinolin-8-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-{[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
ethyl 2-(1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
methyl 3-(furan-2-amido)-1-methyl-5-{[(3-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3,4-dimethoxyphenyl)-2-{methyl[2-(piperidin-1-yl)ethyl]amino}acetic acid
4-{[(butan-2-yl)(3-phenylprop-2-yn-1-yl)amino]methyl}benzoic acid
(1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}azepan-2-yl)methanol
3-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}-N-methylpropanamide
1-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-cyclohexyl-3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propanamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]pyrrolidin-3-yl]methanol
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
7-(2-hydroxyethyl)-2-[2-(3-methoxyphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N3-(1H-1,3-benzodiazol-2-ylmethyl)-N5-cycloheptyl-1-cyclopropyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
N-(2-hydroxypyridin-3-yl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
3-chloro-N-cyclopentyl-4-({1-[2-(furan-2-yl)-2-oxoacetyl]piperidin-4-yl}oxy)benzamide
6-(1-ethyl-5-oxopyrrolidine-3-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-methyl-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2,3-dimethyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]-1H-indole-7-carboxamide
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2-(pyrrolidin-1-yl)propanamide
2-oxo-8-[3-(1H-pyrazol-4-yl)propanoyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[(5-chloro-2,3-dimethoxyphenyl)methyl]azetidin-3-ol
{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}[(3,5-dimethoxyphenyl)methyl](2-methoxyethyl)amine
(3S,4S)-1-[(5-methylfuran-2-yl)methyl]-4-[4-(9H-purin-6-yl)piperazin-1-yl]pyrrolidin-3-ol
methyl (2S,4S)-4-(2-phenylbenzamido)-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
1-(cyclopropylmethyl)-5-(5-methylthiophene-2-carbonyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-methyl-2-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyridine-3-carboxamide
1-(5-chloropyridin-2-yl)-4-[2-(dimethylamino)ethyl]-1,4-diazepan-6-ol