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1-methyl-4-[2-(5-methylpyridin-3-yl)pyridine-4-carbonyl]piperazine
1-{[2-(3,4-dimethoxyphenyl)-8-methylquinolin-3-yl]methyl}piperidin-3-ol
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(3-methylphenyl)acetamide
5-cyclopropyl-N-[3-(morpholin-4-yl)propyl]-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
3-(1H-imidazol-1-ylmethyl)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]benzamide
(3S,4S)-1-(2-ethylbenzoyl)piperidine-3,4-diol
{1-[(2,7-dimethyl-1H-indol-3-yl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
methyl 7-oxo-9-(thiophen-3-ylmethoxy)-3-(2,4,5-trifluorobenzoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(1-methyl-1H-indol-5-yl)methyl]pyrrolidin-3-yl]methanol
methyl(2-phenylpropyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
4-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]-2-methoxypyridine-3-carbonitrile
2-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-6-methylpyridin-3-ol
4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
1-[(4aR,8aR)-4a-hydroxy-7-[(2-methoxypyridin-3-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
2-(2-oxo-1,3-oxazolidin-3-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]acetamide
1-methyl-N-[(1S)-1,2,3,4-tetrahydronaphthalen-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
N-[2-(4-chlorophenyl)-2-(pyrrolidin-1-yl)ethyl]-4-propylpyrimidine-5-carboxamide
2-[4-({2,4-dimethyl-5-[(4-methylpiperidin-1-yl)methyl]phenyl}methyl)morpholin-3-yl]acetic acid
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-cycloheptyl-1H-1,2,3-triazole-4-carbonyl)piperazine
2-(4-benzyl-3-butyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
4-(1H-pyrazol-4-yl)-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]butan-1-one
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(piperidin-1-yl)ethan-1-one
2-{1-cyclohexyl-5-[2-(phenylamino)pyrimidin-5-yl]-1H-1,2,4-triazol-3-yl}acetamide
2-amino-6-{2-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
2-{4-[2-(dimethylamino)ethoxy]-3-ethoxyphenyl}-1H-1,3-benzodiazole-6-carboxylic acid
1-[4-(3-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenoxy)piperidin-1-yl]-2,2-diphenylethan-1-one
3-(2-{[(4-ethyl-1,3-thiazol-2-yl)methyl]amino}propyl)-3,4-dihydroquinazolin-4-one
methyl(2-phenoxyethyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-fluorophenyl)methyl]benzamide
4-(1H-imidazol-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
4-{[(4aR,8aR)-4a-hydroxy-7-(2-methoxyacetyl)-decahydro-2,7-naphthyridin-2-yl]methyl}benzonitrile
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-4-fluorobenzamide
3-{[4-(2,2-dimethylpropanoyl)piperazin-1-yl]methyl}-7-methoxy-1,2-dihydroquinolin-2-one
4-(3-{[(4-fluorophenyl)methyl]amino}benzoyl)-1λ6-thiomorpholine-1,1-dione
4-(2-hydroxy-5-methylbenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
methyl 4-[({2-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-oxopyrrolidin-2-yl]ethyl}amino)methyl]benzoate
3-ethoxy-1-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propan-1-one
7-(3-phenoxybenzenesulfonyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
1-cycloheptyl-5-(1,2-oxazolidine-2-carbonyl)piperidin-2-one
N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N-butyl-1-cyclohexyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
[(3R,4R)-1-[2-(methylsulfanyl)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{1-[(3-chloro-5-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
3-fluoro-N-[(2R,3R)-1'-[(2-hydroxy-5-methoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
5-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-2H-1,2,3,4-tetrazole
3-[(3R,4S)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
3-{[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]sulfamoyl}-N-propylbenzamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,3,5-tetramethylpyrazolo[1,5-a]pyrimidin-7-amine