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1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carboxamide
N-{7-[3-(dimethylamino)pyrrolidine-1-carbonyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazol-5-yl}cyclohexanecarboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-methylthiophene-2-carboxamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1,2-oxazole-3-carboxamide
2-(4-oxo-3,4-dihydrophthalazin-1-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(6-methoxypyrimidin-4-yl)piperazin-2-one
(1S,5R)-6-(cyclopropylmethyl)-3-(1H-imidazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)spiro[2.3]hexane-1-carboxamide
6-ethyl-2-methyl-N-[2-(methylsulfamoyl)ethyl]quinoline-4-carboxamide
2-(dimethylamino)-N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(4-methylphenyl)acetamide
2-[5-(3-ethyl-4-methyl-1H-pyrazol-5-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-3-yl]pyridine
1-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidine-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}bis(prop-2-en-1-yl)amine
2-{4-[(5-ethylfuran-2-yl)methyl]-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl}ethan-1-ol
ethyl 4-[(4-methoxyphenyl)methyl]-1-(thiophene-3-carbonyl)piperidine-4-carboxylate
[(2S,6S)-11-methoxy-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
4-[2-(methylsulfanyl)ethyl]-5-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-methyl-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
ethyl 4-{[1-(4-cyclopentaneamidophenyl)piperidin-4-yl]amino}piperidine-1-carboxylate
2-[3,5-bis(trifluoromethyl)phenyl]-4-hydroxy-N-(2-methoxyethyl)-N-methylpyrimidine-5-carboxamide
(3S,5S)-1-(3-fluoro-4-methylbenzoyl)-5-(morpholine-4-carbonyl)piperidine-3-carboxylic acid
4-ethyl-6-{4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-1-yl}pyrimidine
6-methyl-N-(oxan-4-ylmethyl)-2-phenylpyrimidin-4-amine
3-(2-fluorophenyl)-N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(morpholine-4-carbonyl)pyrrolidin-3-yl]methanol
N-(2,3-dihydro-1H-inden-2-yl)-1-methyl-1H-indole-6-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
{1-[7-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-2H-[1,3]dioxolo[4,5-g]quinolin-6-yl]piperidin-3-yl}methanol
3-[(7-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine
3-(benzyloxy)-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(oxolan-2-ylmethyl)acetamide
4-fluoro-N,3-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
2-(4-{2-[(2-methylphenyl)methoxy]phenyl}-1H-1,2,3-triazol-1-yl)ethan-1-amine
5-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl}-3-(propan-2-yl)-1,2-oxazole
3-{3-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5,6-dimethyl-1,2-dihydropyridin-2-one
1-benzyl-2-(2-methoxyethanesulfonyl)-5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-imidazole
N-(2-hydroxybutyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-benzyl-6-(cyclopropylmethoxy)-4-(3,4,5-trimethoxybenzoyl)-1,4-diazepan-2-one
4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]piperidin-3-ol
(1-{5-[(thian-4-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-yl)methanol
1-(4-methoxyphenyl)-2,2-dimethyl-N-[(3-methylpyridin-2-yl)methyl]cyclopropane-1-carboxamide
N-[2-(methylsulfamoyl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
2-methyl-3-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]-1,8-naphthyridine
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-(2-methoxyphenoxy)ethan-1-one
4-(6-methylpyridine-3-carbonyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol