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1-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
methyl 5-({[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}amino)-1-[2-(1H-indol-3-yl)ethyl]-3-(2-methoxyacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-{[2-(trifluoromethyl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
methyl N-(2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-oxoethyl)carbamate
N-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
[1-(1,3-benzothiazol-2-yl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[1-(3-methylpyridin-2-yl)propyl]acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methanol
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyl-3-(pyrrolidin-1-yl)propanamide
1-methyl-1'-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-benzyl-N-(cyclopropylmethyl)-2-{1-ethyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}acetamide
1-(cyclopropylmethyl)-N-ethyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(3-ethyl-3-hydroxypiperidin-1-yl)-N-(2-hydroxyethyl)pyridine-2-carboxamide
7-[2-(morpholin-4-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[(4-chlorophenyl)methyl]amine
3-({1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)propanamide
N-methyl-5-[(methylsulfanyl)methyl]-N-(pyrazin-2-ylmethyl)furan-2-carboxamide
2-(5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)phenol
1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-4-phenoxypiperidine-4-carboxylic acid
N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
7-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[4-methyl-3-(thiophen-2-yl)-1H-pyrazol-1-yl]acetamide
(3S)-1-{5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}pyrrolidin-3-ol
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(piperidin-3-yl)benzamide
3-({4-[3-(4-ethylpiperazin-1-yl)-3-oxopropyl]piperidin-1-yl}methyl)benzonitrile
1-(4-methoxy-2,3-dimethylphenyl)-2-[5-(methoxymethyl)furan-2-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
1-{1-[3-(methylsulfanyl)propyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
(1R,5S)-6-[(1-ethyl-1H-indol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
ethyl 2-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]amino}acetate
methyl[(1-methyl-1H-pyrazol-4-yl)methyl]{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
4-({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-2-yl}methyl)morpholine
ethyl({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
methyl 4-({3-[(furan-2-ylformamido)methyl]piperidin-1-yl}methyl)benzoate
(1R,9aR)-1-({[2-(2-methoxyphenyl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-cyclopropyl-9-(2-methylpyrimidin-4-yl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(2R,4R,6S)-2-(4-chlorophenyl)-6-(5-methyl-1-propyl-1H-pyrazol-4-yl)oxan-4-yl]acetamide
5-(naphthalen-2-ylmethyl)-5-[3-oxo-3-(piperidin-1-yl)propyl]pyrrolidin-2-one
N-[2-(dimethylsulfamoyl)ethyl]-2-methoxyquinoline-4-carboxamide
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-2-(propan-2-yloxy)propanamide
2-[3-(azetidine-1-carbonyl)benzenesulfonamido]-N-cyclopropylacetamide
3-[(2-fluorophenyl)methyl]-5-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-1,2,4-oxadiazole
1-[4-(4-fluorophenoxy)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
2-(oxolan-3-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(4aS,7aR)-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[4-(4-methoxybenzoyl)piperazin-1-yl]propan-1-one