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1-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)ethan-1-one
N-phenyl-3-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-4-yl}propanamide
3-[(6-hydroxy-1,4-oxazepan-4-yl)methyl]-5,6,7-trimethoxy-1,2-dihydroquinolin-2-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-oxo-1-phenylpyrrolidine-3-carboxamide
(1R,5R)-3-(2,6-difluorobenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-methyl-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-(oxan-4-ylmethyl)butanamide
N-[2-(benzylsulfanyl)ethyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine
2-(4-fluorophenyl)-N-{1-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]-1H-pyrazol-5-yl}acetamide
4-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-5-phenyl-2-(pyridin-4-yl)pyrimidine
N-{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
7-(1,3-benzothiazol-2-yl)-4-propyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
[(3R,4R)-1-(1-methyl-1H-indole-3-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[5-(3-chlorophenoxymethyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methanamine
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-[2-(1,3-thiazol-2-yl)ethyl]propanamide
2-(3-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}pyrazolo[1,5-a]pyrimidin-6-yl)ethan-1-ol
(4-{[(7-chloroquinolin-4-yl)(methyl)amino]methyl}oxan-4-yl)methanol
1-(prop-2-en-1-yl)-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]pyrrolidin-2-one
2-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-(4-hydroxypiperidin-1-yl)-2-[4-(4-{[2-(3-methoxyphenyl)ethyl]amino}piperidin-1-yl)phenyl]ethan-1-one
2-({3-cyclopropyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1-(2-methoxyethyl)-1H-imidazole
(5S,9aS,9bS)-5-(1-ethyl-1H-imidazol-2-yl)-2-[(5-methylfuran-2-yl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[(4-methoxyphenyl)methyl]-N-[3-(pyridin-3-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
(1S,3R)-N1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(4-methoxyphenyl)ethyl]piperidine-3-carboxamide
4-(4-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}piperidin-1-yl)-1λ6-thiane-1,1-dione
1-(2-methyl-1,3-thiazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-7-acetamido-2-(2-methoxyphenyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-4-phenylbutan-1-one
[3-(prop-2-en-1-yl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-3-yl]methanol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
4-{1-[6-(2-methylpyrrolidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}morpholine
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methylpyridine
(1R,5R)-6-(cyclopropylmethyl)-3-(thiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(1H-pyrazole-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
N-cyclopropyl-1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}piperidine-4-carboxamide
[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})methylamine
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(1-methyl-1H-indol-6-yl)methyl]pyrrolidin-3-yl]methanol
N,N,7-trimethyl-3-({[(3,4,5-trimethoxyphenyl)methyl]amino}methyl)quinolin-2-amine
1-(1-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-4-yl}ethyl)-4-methylpiperazine
5-methyl-N-{[8-(propan-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1,3,4-oxadiazol-2-amine
1-cyclopropyl-5-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}piperidin-2-one
6-[2-(tert-butylsulfamoyl)phenyl]-N,N-dimethylpyridine-3-carboxamide
N-benzyl-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}propanamide
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
6-(8-methoxy-2-methylquinolin-5-yl)-N,N-dimethylpyrazine-2-carboxamide
2-{2-[3-(methoxymethyl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione