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(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(butane-1-sulfonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(6,8-difluoroquinolin-4-yl)aniline
2-methoxy-4-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
N-(4-methyl-2-{2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamido}phenyl)benzamide
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidine-4-carbonitrile
5-ethyl-N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-methylpyrimidin-4-amine
(2S,4R)-4-amino-1-(6-oxo-1,6-dihydropyridine-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]({6-methyl-2-[(2-methylphenyl)methoxy]quinolin-3-yl}methyl)amine
5-{2-[4-(2-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-3-propylimidazolidine-2,4-dione
4-(1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidine-4-carbonyl)morpholine
N-[(2R,3R)-2-methoxy-1'-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-[(3S,5S)-1-ethyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-6-fluoro-4-hydroxyquinoline-3-carboxamide
6-(methoxymethyl)-N-methyl-N-(2-phenoxyethyl)pyrimidin-4-amine
5-({[1-tert-butyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]methyl}sulfanyl)-1,3,4-thiadiazol-2-amine
2-amino-4-(3-chloro-4-fluorophenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N,N-dimethylpropanamide
5-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
7-(cyclobutylmethyl)-2-(2-methyl-1,3-thiazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclohexyl-3-[(3S)-3-ethylmorpholine-4-carbonyl]-N-methylpyridin-2-amine
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(prop-2-en-1-yl)acetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2,3-dimethoxyphenyl)methyl]propanamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(4-fluorophenyl)-1,4-diazepane
2-chloro-4-fluoro-N-{[8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
6-{4-[3-(dimethylamino)-2,2-dimethylpropyl]piperazin-1-yl}pyridine-3-carbonitrile
6-methyl-2-{[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
4-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-2,2-dimethylmorpholine
4-ethyl-N,N-dimethyl-6-[4-(propan-2-yl)piperazin-1-yl]pyrimidin-2-amine
2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-N-(2-fluoro-4-methylphenyl)propanamide
N3-benzyl-N5-tert-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(3aS,6aS)-2-[(6-methylpyridin-2-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-ethoxy-N-(2-methoxy-5-phenylphenyl)piperidine-1-carboxamide
4-(2-fluorophenoxy)-1-(3-methylbenzoyl)piperidine-4-carboxylic acid
4-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
[3-benzyl-1-(5-fluoro-2-methylbenzenesulfonyl)piperidin-3-yl]methanol
2-(1H-imidazol-1-yl)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
1-{[(3-fluorophenyl)methyl]carbamoyl}-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(2-{5-[(E)-2-(2-methoxyphenyl)ethenyl]-4-phenyl-1H-imidazol-1-yl}ethyl)acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylphenol
N-[4-(1-methyl-1H-indol-2-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]methanesulfonamide
2-({4-[3-(1,3-benzothiazol-2-yl)propanoyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)-N,N-diethylacetamide
N-[(3-chlorophenyl)methyl]-3-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]propanamide
N-(4-fluorophenyl)-2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidine-6-carboxamide
3-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-[(2-hydroxyethyl)(methyl)amino]acetamide
N-cyclopropyl-1-{7-methyl-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}piperazine-2-carboxamide
1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethan-1-amine
4-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-1-[(5-methyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole
N-(2-methoxyethyl)-N,5-dimethyl-4-[(2-phenylethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide