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[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-butyl-3-cyclopropyl-5-[(2,4-difluorophenyl)methyl]-1H-1,2,4-triazole
N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
9-{[3-(2-aminoethyl)phenyl]methyl}-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
4-[2-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzene-1-sulfonamide
7-(5-chloropyridin-2-yl)-4-[(2,4-dimethoxy-3-methylphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,3-difluorophenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
N-(cyclobutylmethyl)-4-methoxy-N-(oxolan-2-ylmethyl)-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
1-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
N-(4-oxo-4H-chromen-6-yl)-2-[2-(pyridin-2-yl)ethyl]piperidine-1-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
4-hydroxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]benzamide
(3S,4R)-4-(3-fluorophenyl)-1-[2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]pyrrolidine-3-carboxylic acid
N-methyl-N-(1H-pyrazol-3-ylmethyl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
N-(1-phenylethyl)-3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-(2H-1,3-benzodioxol-4-ylmethyl)-3-(naphthalene-1-carbonyl)piperidine
1-methyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole-6-carboxamide
2-(2-methoxyethyl)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[3-(2-phenylethyl)piperidin-1-yl]ethan-1-one
2-methoxy-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
N-[2-(1H-imidazol-1-yl)ethyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
3-amino-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1H-1,2,4-triazole-5-carboxamide
N-[2-(propan-2-yloxy)ethyl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(3-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-4-oxo-N-[4-(pentyloxy)phenyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
6-{2-[bis(propan-2-yl)carbamoyl]phenyl}pyrazine-2-carboxylic acid
(2H-1,3-benzodioxol-4-ylmethyl)(methyl)[(3-phenyl-1H-pyrazol-4-yl)methyl]amine
N-[1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]pyrimidin-2-amine
5-phenyl-3-[3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-1,2,4-triazine
methyl (2S,4R)-4-(dimethylamino)-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}pyrrolidine-2-carboxylate
9-(2-methoxyethyl)-1-methyl-4-(pyrimidin-2-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N,5,7-trimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-{[methyl(1-methylpiperidin-4-yl)amino]methyl}-4-(pyrazin-2-yl)phenol
4-(4-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]amino}piperidin-1-yl)-N,N,6-trimethylpyrimidin-2-amine
N,1-dimethyl-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,6-dihydropyridazine-3-carboxamide
N-benzyl-5-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[4-(1-cyclohexanecarbonylpyrrolidine-2-carbonyl)-1,4-diazepan-1-yl]-2,2,2-trifluoroethan-1-one
4-(2,4-dioxoimidazolidin-1-yl)-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]benzamide
2-methyl-6-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
(2E)-1-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-3-(furan-2-yl)prop-2-en-1-one
1-(4-methanesulfonyl-1,4-diazepan-1-yl)-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-cyclohexyl-N-[1-(furan-2-carbonyl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
dimethyl({[2-(2-methylphenoxy)pyridin-3-yl]methyl}sulfamoyl)amine
3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-({[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl](methyl)amino}methyl)phenol
4-(1-{3-[(1-methylpiperidin-4-yl)oxy]propyl}-1H-imidazol-2-yl)pyridine