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2,6-dihydroxy-N-[1-(4-methanesulfonylphenyl)propyl]benzamide
(5S)-5-[({[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-3-ylmethyl)amino)methyl]pyrrolidin-2-one
N-ethyl-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
7-chloro-4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-tert-butyl-N-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
N-{3-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]-3-oxopropyl}-4-fluorobenzamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-ol
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-[(2-fluorophenyl)methyl]-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-3-yl}propanamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-[(4-methylphenyl)amino]-2-phenylpropanamide
6-cyclopropyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}pyrimidin-4-amine
1'-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(dicyclopropylmethyl)({[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-[(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]phenol
N-[(5-methylpyrazin-2-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
(2R,6S)-4-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2,6-dimethylmorpholine
5-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1H-indole
3-chloro-N-cyclopropyl-N-{[6-(2,5-dimethoxyphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
4-methoxy-3,5-dimethyl-2-{[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]methyl}pyridine
1-(7-{[4-(pyridin-2-ylmethyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(thiophen-2-yl)ethan-1-one
3-bromo-N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
1-(carbamoylmethyl)-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
7-(1-benzothiophen-3-yl)-4-(1H-imidazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-({8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-2-methoxybenzoic acid
1-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-1,4-diazepan-1-yl)ethan-1-one
1-cycloheptylpiperidin-3-amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-3-ethyl-1-methyl-N-[2-(piperidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
7-cyclohexyl-2-(2-phenoxyacetyl)-2,7-diazaspiro[4.5]decan-6-one
4-(cyclopropylmethyl)-1-(1,3-dihydroxypropan-2-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
N,N-dimethyl-2-({[2-(methylsulfanyl)pyrimidin-4-yl]amino}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(3-methylphenyl)acetamido]methyl}benzoate
N-[(3S,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-propylpyrrolidin-3-yl]acetamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-(1H-indol-4-ylmethyl)propanamide
4-(1-ethylpiperidin-4-yl)-11-(2-methylbenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
[5-(1-{[5-(2-fluorophenyl)furan-2-yl]methyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-5-phenyl-1,2-oxazole-3-carboxamide
N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}-1H-1,2,3-triazole-5-carboxamide
4'-butyl-1-(2,2-dimethylbutanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
({5-[1-(1-cyclopropyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-benzoyl-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-[1-(2-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
3-(5-methylthiophen-2-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
7-(5-chloropyridin-2-yl)-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(3-fluorophenyl)-N-[3-(1H-indol-1-yl)propyl]-1,2,4-triazin-3-amine
ethyl 2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]acetate
4-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,2-dimethylpiperazine
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
4-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide