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ethyl 1-[(4-methoxy-2-methylphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
methyl (2S,4S)-1-[1-(2-phenylethyl)piperidin-4-yl]-4-[2-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxybenzoyl)piperidine
4-[5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)furan-2-yl]-2-methylbut-3-yn-2-ol
9-methoxy-7-(3-methoxyphenyl)-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-methoxy-4-({[(2-methoxyphenyl)methyl](methyl)amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-3-(1,2-oxazolidin-2-yl)-N-(pyridin-4-ylmethyl)propanamide
3-(2-methylphenyl)-1-[4-(pyridin-2-yl)pyrimidin-2-yl]pyrrolidin-3-ol
3-bromo-N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
1-{3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]phenyl}ethan-1-one
4-{4-[4-(4-methylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(4-cyclopentyl-3-oxopiperazin-1-yl)-N-(2,4-dimethoxyphenyl)-3-oxopropanamide
6-(5-acetylthiophene-3-carbonyl)-1-(cyclopropylmethyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
4-[6-(thiomorpholin-4-yl)pyridazin-3-yl]phenol
N5-ethyl-N6,N6-dimethyl-N5-[2-(1H-pyrazol-1-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-ethyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1H-pyrazole-4-carboxamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-[2-(methylsulfanyl)benzoyl]-1,4-diazepan-2-one
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)thieno[2,3-b]pyridine-2-carboxylate
N-(1-carbamoylcycloheptyl)-5-(3-methoxyphenyl)furan-2-carboxamide
2-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-1-(3,5-dimethoxyphenyl)ethan-1-ol
3-(1H-1,3-benzodiazol-1-yl)-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}propanamide
[(5-methyl-1,2,4-oxadiazol-3-yl)methyl][(4-methyl-1H-imidazol-5-yl)methyl](propan-2-yl)amine
(1S,9R)-11-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(1-propylpiperidin-3-yl)methyl]butanamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
(3R,5S)-5-(3-fluorophenoxymethyl)-N,1-bis(2-phenylethyl)piperidine-3-carboxamide
N-cyclohexyl-N-ethyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-benzyl-9-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(4-chloro-1H-pyrrole-2-carbonyl)-6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline
(1S,5R)-6-{4-[(2-fluorophenyl)methoxy]benzoyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
5-(1H-imidazol-1-yl)-N-(2-methoxyethyl)furan-2-carboxamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyrimidine-3-carboxamide
2-({4-[6-(cyclopentylamino)pyridazin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
1-cyclohexyl-4-[2-(4-methoxyphenyl)acetyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
3-[({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)methyl]pyrrolidin-3-ol
1-(2-methylphenyl)-4-{1-[2-(trifluoromethyl)benzoyl]piperidin-3-yl}piperazine
2-[4-methoxy-3-(methoxymethyl)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-cyclopentylpiperazin-2-one
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-[4-(methylsulfanyl)phenyl]ethan-1-one
1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine-4-carboxamide
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-[(3-methylphenyl)methyl]pyrrolidine-2-carboxamide
1-methyl-4-{[6-(trifluoromethyl)pyridin-3-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
3-(4-chlorophenyl)-1-[4-(2-methoxyethyl)piperazin-1-yl]-3-phenylpropan-1-one
2-({2-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
3-[(3-methoxyphenyl)methyl]-8-[(4-methyl-1H-imidazol-2-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(3-chlorophenyl)phenyl]-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}urea
N-({8-[(2,4-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1-methyl-1H-pyrazole-3-carboxamide