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(3R,4R)-3-methyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
N-(2,3-dihydro-1H-inden-2-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-chloro-4-({4-[(4-fluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenol
methyl 5-[2-(5-amino-1,3,4-thiadiazol-2-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
2-(3-methoxypropyl)-9-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-(2-chlorophenyl)-4-({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(1-methyl-1H-indol-6-yl)methyl]piperazin-2-one
4-{[1-(but-3-enoyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
2-(3,4-dimethylphenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
N-{1-[({[3-(1H-pyrazol-1-yl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-2H-1,3-benzodioxole-5-carboxamide
1,3-dimethyl-N-{2-[3-(thiomorpholin-4-ylmethyl)phenoxy]propyl}-1H-pyrazole-5-carboxamide
(3R)-1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
1-(4,7-dimethylquinazolin-2-yl)-N-[(2-methoxynaphthalen-1-yl)methyl]piperidine-4-carboxamide
ethyl 4-{1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
4-(1-cyclopentyl-1H-imidazol-2-yl)-2-ethylpyrimidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1H-imidazole-2-carboxamide
N-[1-(1-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
1-[2-methoxy-4-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
8-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2-{1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
7-[2-(4-chloro-3,5-dimethylphenoxy)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-({1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(4aS,8aR)-2-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-decahydroisoquinoline
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]propan-1-one
2-{[(4-ethoxyphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-(1-hydroxy-2-methylpropan-2-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-cyclopropyl-N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
3-benzyl-5-(methanesulfonylmethyl)-1H-1,2,4-triazole
4-[2-(1H-imidazol-4-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-fluoro-N-({8-[(2,4,6-trimethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
7-(5-chloropyridin-2-yl)-9-methoxy-4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{3-methyl-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl}acetic acid
3-({[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]carbamoyl}methyl)-1,2,3-oxadiazol-3-ium-5-olate
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidine
methyl 4-({[(3R,5S)-1-benzyl-5-[(2-methoxyethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
2-(2H-1,3-benzodioxol-5-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
1-(2-{[6-(dimethylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}ethyl)piperidin-2-one
4-[(4-methyl-5-{1-[(6-methylpyridin-2-yl)methyl]piperidin-3-yl}-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carbonyl}pyridine
3-(but-2-yn-1-yl)-5-{1-[(2-chlorophenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]imidazolidine-2,4-dione
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N,N-diethylpiperidine-3-carboxamide
2-methoxy-4-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-4-(pyridin-2-yl)piperazine
(4aS,8aR)-6-(2-amino-6-methoxypyrimidin-4-yl)-1-propyl-decahydro-1,6-naphthyridin-2-one
2-cyclopropyl-5-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)-4-(3-methylthiophen-2-yl)-1H-1,2,3-triazole
({4-cyclopropyl-5-[1-(1-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
(5S,9aS,9bS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-cyclopentyl-N-(4-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-cyclopentyl-3-(2-methylphenyl)-3-[2-(2-methylpiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione