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1-[(1,3-dimethylpyrrolidin-3-yl)methyl]-2-(1H-imidazol-4-yl)-1H-imidazole
4-(3-cyclohexyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl)benzoic acid
1-{4-[7-(morpholin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]phenyl}pyrrolidin-2-one
methyl 1-(2-{[benzyl(ethyl)amino]methyl}-6,7-dimethoxyquinazolin-4-yl)piperidine-4-carboxylate
2-methyl-N-{2-[7-(quinolin-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
(1S,5R)-3-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-amine
3-methyl-N-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholin-2-yl}ethyl)but-2-enamide
2-[(2-methoxyethyl)(methyl)amino]-1-[4-(2-phenylethyl)piperidin-1-yl]ethan-1-one
4-(4-methoxyphenoxy)-1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperidine
5-(phenoxymethyl)-N-(2-phenylpropyl)-1H-pyrazole-3-carboxamide
(morpholin-2-ylmethyl)({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
2-{2-[({[(2R,3R,5S)-2-(4-chlorophenyl)-1-ethyl-5-(hydroxymethyl)-5-methylpyrrolidin-3-yl]methyl}amino)methyl]phenoxy}ethan-1-ol
N-(1-benzofuran-2-ylmethyl)-1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-amine
1-methyl-4-({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
(1S,6R)-3-[(3-chloro-4-fluorophenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane
4-benzyl-3-ethyl-1-(2-methoxybenzoyl)-1,4-diazepan-5-one
4-[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(4-fluorophenyl)ethyl)piperidine-1-carbonyl]pyridin-1-ium-1-olate
1-[2-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
3-methyl-1-{3-[(2-methylpiperidin-1-yl)methyl]phenyl}-3-[2-(pyridin-2-yl)ethyl]urea
7-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-2-oxa-7-azaspiro[4.5]decane
1-methyl-4-{5-[4-(1,2,3-thiadiazol-4-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}piperidine
N-methyl-N-[2-(morpholin-4-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
3-[3-methyl-1-(2-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-indazole
N-(2-{7-[(3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-[(4-cyanophenyl)methyl]-2-(dimethylamino)-2-(2-methylphenyl)acetamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{3-[methyl(phenyl)amino]propyl}propanamide
6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2-dihydropyridin-2-one
ethyl 4-[3-({[2-(cyclohex-1-en-1-yl)ethyl]amino}methyl)-6,7-dimethoxyquinolin-2-yl]piperazine-1-carboxylate
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[3-(3-fluorophenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-(furan-2-ylmethyl)-N-methylacetamide
2-amino-3-ethyl-N-(2,2,2-trifluoroethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-(4-{4-[(2-methoxyethyl)amino]piperidin-1-yl}phenyl)-2,4-dimethylbenzamide
3-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)-1-phenylpropan-1-ol
1-(3-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
1-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]-N,N-dimethylpyrrolidin-3-amine
(4-phenyl-5-{[1-(pyrimidine-5-carbonyl)piperidin-4-yl]methyl}-4H-1,2,4-triazol-3-yl)methanol
N-[3-(2-fluorophenyl)propyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-8-(quinolin-8-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-{[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(4-methylpiperidin-1-yl)-2-[2-(4-phenyl-1H-imidazol-5-yl)phenoxy]ethan-1-one
3-{2-[3-(2-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-(1,2,3-thiadiazole-4-carbonyl)piperidine
5-methyl-N4-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]pyrimidine-2,4-diamine
(2E)-N-({7-[2-(3,4-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
1-cyclopropyl-N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-methoxyethan-1-one
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)amine
N-(dicyclopropylmethyl)-2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methylacetamide