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N-ethyl-3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]benzamide
N-cyclopentyl-1-[(4-methoxyphenyl)methyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3-[1-(1-cyclopropylethyl)-1H-pyrazol-5-yl]urea
2-{2-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}pyridine
5-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
1-(furan-2-yl)-2-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethane-1,2-dione
N,4-dimethyl-N-[2-(4-methylphenoxy)ethyl]-1H-imidazole-5-carboxamide
6-(1-benzylpiperidin-4-yl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(cyclohexylmethyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-[(2S)-1-hydroxybutan-2-yl]-1,3-oxazole-4-carboxamide
3-methyl-8-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
4-{4-[2-(benzyloxy)acetyl]-2-oxopiperazin-1-yl}benzonitrile
N,N-dimethyl-3-(1-methyl-1H-indazol-5-yl)aniline
5-(1-cyclopentylpiperidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-{2-[2-(1H-imidazol-4-yl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-1,3-thiazole-4-carboxamide
3-(3-methoxyphenyl)-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrazole-5-carboxamide
4-[4-(3-methylphenoxy)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(3,4-dimethoxyphenyl)propan-1-one
(furan-2-ylmethyl)({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(prop-2-yn-1-yl)amine
5-({[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-methoxyphenol
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(4-hydroxyphenyl)-N-[(4-methylphenyl)(pyridin-4-yl)methyl]propanamide
N-cyclopropyl-2,3-dimethyl-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-1H-indole-5-carboxamide
2-{3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}ethan-1-ol
(3S,4S)-4-(morpholin-4-yl)-1-[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]pyrrolidin-3-ol
9-methoxy-N-methyl-7-oxo-3-(2-phenoxypropanoyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
ethyl 4-[(pyrazin-2-yl)amino]piperidine-1-carboxylate
4-(1-butyl-1H-imidazol-2-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
1-[(4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]cyclopropane-1-carboxamide
5-methoxy-3-[1-(6-methylpyridin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
4-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-6-methylpyrimidin-2-amine
N-benzyl-1-methyl-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[1-(furan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-3-methyl-1,2-benzoxazole
(3S,4R)-1-(2,5-difluorobenzoyl)-N,N-dimethyl-4-propylpyrrolidin-3-amine
1-[3-(4-fluorophenyl)propanoyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(piperidin-4-yl)piperidine
methyl 3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]benzoate
8-fluoro-N-[2-(pyrrolidine-1-sulfonyl)ethyl]quinoline-2-carboxamide
(2S,4R)-4-amino-1-(6-cyclopropylpyrimidin-4-yl)-N-methylpyrrolidine-2-carboxamide
2-(ethylamino)-N-methyl-N-(thiophen-3-ylmethyl)pyrimidine-5-carboxamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
5-(2,6-dimethylphenoxymethyl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1,2-oxazole-3-carboxamide
1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-{5-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-yl]-3-cyclopropyl-1H-1,2,4-triazol-1-yl}pyridine
N-{[3-methyl-7-(3-methyl-2-oxopentanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-3-carboxamide
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-methyl-N-{1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]-2-phenylethyl}oxane-4-carboxamide
2-[5-(3-phenylpropyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline