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4-(4-acetamido-1H-pyrazol-1-yl)-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]benzamide
2-(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}azetidin-3-yl)pyridine
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(2S,4S)-4-{[(3-chlorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-(1,2-oxazol-3-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
2-chloro-N-{2-[(2-cyclopropyl-4-methylpyrimidin-5-yl)formamido]ethyl}benzamide
3-phenyl-N-{[5-(thiophen-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
5-tert-butyl-N-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,3,4-oxadiazol-2-amine
2-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]-1,2-dihydrophthalazin-1-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[3-(2-fluorophenyl)benzoyl]-1,4-diazepan-5-one
3-fluoro-4-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}benzamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N-ethyl-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
6-(benzyloxy)-1-cyclohexyl-4-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-1,4-diazepan-2-one
7-(cyclohexylmethyl)-6-oxo-N-(prop-2-en-1-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
4-{[1-(3-phenylphenyl)piperidin-4-yl]amino}butan-1-ol
1-(3-chlorophenyl)-4-cyclopentanecarbonyl-5-methylpiperazin-2-one
N-cyclohexyl-4-[(dimethylamino)methyl]-N-(pyridin-2-ylmethyl)benzamide
2-[4-(azepan-1-ylmethyl)phenyl]-6-cyclopentyl-3,4-dihydropyrimidin-4-one
[3-methyl-1-({2-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidin-3-yl]methanol
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
dimethyl({3-[2-(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
1-(3-chlorophenyl)-4-[3-(4-fluorophenyl)propanoyl]piperazin-2-one
5-(2,6-difluorophenoxymethyl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,4-dithiepan-6-amine
2-(carbamoylamino)-N-(isoquinolin-5-ylmethyl)-N-methylacetamide
N-[(3S,4R)-1-[(1-methyl-1H-indol-5-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-methyl-1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazole-4-carboxylic acid
5-(4-phenyl-1,4-diazepane-1-carbonyl)pyrrolidin-2-one
N,N-dimethyl-2-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
4-[2-(1H-imidazol-1-yl)acetyl]-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
1-[(3S,7S)-3-(hydroxymethyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(14),10,12-trien-5-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-{3-[(2-methoxyphenyl)methyl]-5-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
1-(2-methylpropyl)-5-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenylacetamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]propanamide
3-{2-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(3-methoxyphenyl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(3-fluorophenyl)-6,6-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrimidin-2-amine
3-{2-[4-(2-chlorophenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
6,7-dimethoxy-2-(morpholine-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline
8-fluoro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
N,6-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridazin-3-amine
3-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]aniline
3-hydroxy-3-[({[1-(hydroxymethyl)cyclobutyl]methyl}(methyl)amino)methyl]-1-[(3-methylphenyl)methyl]piperidin-2-one
9-{[5-chloro-2-(prop-2-en-1-yloxy)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-[2-(5-methyl-4-{[methyl({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})amino]methyl}-1,3-oxazol-2-yl)phenyl]methanesulfonamide
[(3R,4S)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-{2-[7-(5-chloro-2-methoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-6-methoxy-2,3-dihydro-1H-indol-2-one
methyl 6-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine-3-carboxylate