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2-benzyl-8-(6-hydroxyhexyl)-2,8-diazaspiro[5.5]undecan-3-one
2,6-dimethyl-5-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydropyrimidin-4-one
2-(2-{[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-[4-(1H-pyrazol-3-yl)benzoyl]-1,2-oxazolidin-4-ol
3-methyl-2-(4H-1,2,4-triazol-4-yl)-5-(2,4,6-trimethylphenyl)pyridine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-ol
2-ethyl-1-methyl-4-[(2,3,4-trimethoxyphenyl)methyl]piperazine
{[2-(furan-2-yl)phenyl]methyl}(methyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-N-methylpiperidine-2-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-methoxyethyl)-4-methyl-3-{[(2-methylprop-2-en-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-cyclopropyl-4-methoxy-2-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
1-[4-({4-[4-(furan-2-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-1-yl]ethan-1-one
N-[4-(furan-2-yl)butan-2-yl]-6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-(1H-pyrazol-1-yl)acetamide
1-{[2-(4-chlorophenyl)-7-methoxyquinolin-3-yl]methyl}piperidine-4-carbonitrile
(1R,5R)-6-[(2-aminopyridin-3-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypyrazine
N-{[3-(2,4-dimethoxyphenyl)phenyl]methyl}propanamide
1-[1-ethyl-5-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
4-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-{4-[(1R,3R,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane-8-carbonyl]piperidin-1-yl}ethan-1-one
4-ethyl-5-methyl-6-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-2-amine
2-(4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)quinazoline
(4aS,8aR)-6-[5-(propan-2-yl)pyrimidin-4-yl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
3-{[4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}pyridine
6-(8-methoxyquinolin-5-yl)-4-(4-methylpiperazin-1-yl)quinazoline
2-[2-(1H-imidazol-4-yl)ethyl]-8-(1H-imidazole-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(4-methylpiperazin-1-yl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,3-dihydropyridazin-3-one
N-{[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}cyclopentanamine
2-{[4-(3-methoxyphenyl)-5-(oxan-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(2-oxopyrrolidin-1-yl)-N-(pyridin-3-ylmethyl)propanamide
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-ol
4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-1-(2-methoxyphenyl)piperazin-2-one
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(3,5-dimethyl-1H-pyrazol-4-yl)ethan-1-one
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-methyl-1,3-thiazole-4-carboxamide
N-(7-{6-azabicyclo[3.2.1]octane-6-carbonyl}-1-ethyl-2-(3-methoxyphenyl)-1H-1,3-benzodiazol-5-yl)acetamide
3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-(4-methoxyphenyl)-7-methylquinoline
N-[(3R,4R)-3-hydroxy-1-(6-methylpyridazin-3-yl)piperidin-4-yl]pyridine-2-carboxamide
8-[(3-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl){2-[(4-methylphenyl)sulfanyl]ethyl}amine
(1R,9aR)-1-[({3-[(5-methylpyridin-2-yl)amino]propyl}amino)methyl]-octahydro-1H-quinolizin-1-ol
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methyl-1H-indol-3-yl)ethan-1-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(pyrrolidine-1-carbonyl)piperidine
3-{4,5-dimethyl-1-[5-(methylcarbamoyl)furan-2-yl]-1H-1,3-benzodiazol-2-yl}propanoic acid
4-[(2-chloro-4-ethoxy-5-methoxyphenyl)methyl]-1-phenylpiperazin-2-one
[4-methyl-1-({4-[3-(morpholin-4-yl)propoxy]phenyl}methyl)piperidin-4-yl]methanol
3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
(1R,5R)-6-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane