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[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amine
1-[1-(3-fluoropyridine-4-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
5-(2-chloro-6-fluorophenyl)-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(1-methyl-1H-pyrrol-3-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-(2-methyl-1,3-benzothiazol-5-yl)-6-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-(6-methoxyquinolin-8-yl)-3-(pyrimidin-4-yl)piperidine-1-carboxamide
7-cyclobutanecarbonyl-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-(4-methoxypyrimidin-2-yl)-2,5-diazabicyclo[2.2.1]heptan-3-one
methyl (2S,4S)-4-{[(2-ethoxyphenyl)carbamoyl]amino}-1-methylpyrrolidine-2-carboxylate
(2R)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]oxolane-2-carboxamide
3-[2-(6-methoxynaphthalen-2-yl)ethyl]-1λ6-thiolane-1,1-dione
methyl 1-[(3S,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-(cyclohexylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-(2-phenoxyethyl)-4-(5-propyl-1,2-oxazole-4-carbonyl)piperazine
9-benzoyl-2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-[(1R,5R)-6-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2E)-1-[4-(2-phenylpyrimidin-4-yl)piperidin-1-yl]-3-(pyridin-4-yl)prop-2-en-1-one
(3R,4S)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(3-methoxyphenyl)pyrrolidin-3-amine
1,5-dimethyl-4-({8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decan-1-yl}methyl)-1H-pyrrole-2-carbonitrile
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-methyl-1H-pyrazole-4-carboxamide
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-6-ethyl-2-methylquinoline-4-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(quinoxaline-6-carbonyl)piperidine-3-carboxylate
N-{[(2S,4S)-4-fluoro-1-{[5-(1,2-oxazol-3-yl)thiophen-2-yl]sulfonyl}pyrrolidin-2-yl]methyl}acetamide
(2S)-2-amino-4-[1-cyclohexyl-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-5-yl]butanoic acid
N-[(3R,4S)-1-acetyl-4-cyclopropylpyrrolidin-3-yl]-3-chloro-4-methylbenzene-1-sulfonamide
1-{1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}propan-1-ol
1-(1,3-benzothiazol-2-yl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(2,5-dimethylbenzoyl)-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-{4-[(propan-2-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2,5-dimethoxy-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
(3S,4R)-1-[6-(methoxymethyl)pyrimidin-4-yl]-4-methylpiperidine-3,4-diol
8-[5-(1H-imidazol-4-ylmethyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl]quinoline
8-[4-hydroxy-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)furan-3-carboxamide
1-(pyrrolidin-1-yl)-N-(quinolin-2-ylmethyl)cyclopentane-1-carboxamide
(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-{[(3-chlorophenyl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
N-{[8-({4-[methyl(phenyl)amino]phenyl}methyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}furan-2-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-4-yl]propanamide
4-{5-[1-(1-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-2-yl]thiophene-2-carbonyl}morpholine
3-methoxy-N-[4-(3-methoxyphenyl)phenyl]piperidine-1-carboxamide
(3S)-1,3-dimethyl-4-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
4-[(3-fluorophenyl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)-3-oxopiperazine-1-carboxamide
5-{4-[(2-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
methyl 4-{[4-(3-hydroxyphenyl)piperidine-1-carbonyl]amino}-3-methylbenzoate
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-1H-indole-4-carboxamide
N-(1H-indol-2-ylmethyl)-N'-[2-(methylsulfanyl)phenyl]butanediamide
9-oxo-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraene-10-carboxamide