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2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-[2-methoxy-4-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-cyclopropyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]pyrimidine-5-carboxamide
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-phenylbutanamide
N-benzyl-1-[1,3-dioxo-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-ethylpiperidine-4-carboxamide
3,5-dimethyl-4-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrrole-2-carboxylic acid
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-(2-phenylethyl)-5-(1H-pyrazol-3-yl)-1,2,4-oxadiazole
3-{2-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-thiazolidine-2,4-dione
[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methanol
5,5-dimethyl-3-{2-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidine-2,4-dione
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-{[(4-fluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
N-[(2,6-difluorophenyl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]methanesulfonamide
6-[(2,6-difluorophenyl)methyl]-N-(2-methoxyphenyl)-6-azaspiro[2.5]octane-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
N-{2-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}oxolane-2-carboxamide
2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-5-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]benzamide
2-(3-fluoro-4-hydroxyphenyl)-1-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}ethan-1-one
N-[(1R,2S)-2-phenylcyclohexyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
3-(1,2-oxazolidin-2-yl)-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
7-(cyclobutylmethyl)-2-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
({4-ethyl-5-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-ethyl-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-(2-methylprop-2-en-1-yl)propanamide
1-({4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
(3S,4S)-3-hydroxy-4-[methyl({5-[4-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl})amino]-1λ6-thiolane-1,1-dione
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-6-oxo-N-(oxolan-2-ylmethyl)-1,6-dihydropyrimidine-5-carboxamide
(2S)-N-(3-hydroxypropyl)-1-methyl-N-[(5-methylthiophen-2-yl)methyl]pyrrolidine-2-carboxamide
3-amino-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-[2-(diethylamino)ethyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-chloro-9-methyl-3-({methyl[3-(phenylsulfanyl)propyl]amino}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
2-(2-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)acetic acid
4-[4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine-1-carbonyl]morpholine
(2S)-2-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}pentanediamide
3-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-1-[(3-hydroxypiperidin-3-yl)methyl]urea
(3aS,6aS)-2-(oxan-4-yl)-5-[(trimethyl-1H-imidazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(5-chloropyridin-2-yl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-[4-(2-methylpropoxy)phenyl]-3-[2-(pyridin-3-yl)ethyl]urea
N-[1-(1H-imidazol-1-yl)butan-2-yl]-1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-methyl-6-[3-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-(2-methoxyphenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-4-carboxamide
2-amino-N-[(2,4-difluorophenyl)methyl]-4-phenylpyrimidine-5-carboxamide
N-(butan-2-yl)-7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-methyl-N-(2-phenoxyethyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
1-[(3-fluorophenyl)methyl]-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
N'1-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}cyclopropane-1,1-dicarboxamide
(3S,4S)-1-(3-fluoropyridin-2-yl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-{[4-(1-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-(2-fluorophenyl)ethyl)piperidin-1-yl]methyl}-6-methoxyphenol
(1R,2S,9R)-11-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one