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N-{1-[1-(quinolin-8-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
1-[(3-methylpyridin-2-yl)methyl]-4-(2-phenylpropyl)piperazine
N-(2-{1-[(6,8-dimethyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-2-yl}ethyl)acetamide
N-[1-({[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-3-phenoxypropanamide
2-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3,5-dimethoxyphenyl)methyl]-3-[(4-fluorophenyl)formamido]propanamide
1-(3-methoxypyrazin-2-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane
5-[(4,4-difluoropiperidin-1-yl)methyl]-2-(pyridin-2-yl)pyrimidine
2-(3,4-difluorophenyl)-N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
2-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-1-(morpholin-4-yl)ethan-1-one
N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
(3R,4R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
6-[(3-fluorophenyl)methoxy]-4-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
3-(hydroxymethyl)-N-(6-methylpyridin-3-yl)piperidine-1-carboxamide
4-[3-(piperidin-4-ylmethyl)benzoyl]-2-(trifluoromethyl)morpholine
1-{2-[(3,5-dimethoxyphenyl)formamido]ethyl}-N-(2-methoxyphenyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-methoxypropyl)-4-(naphthalen-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(3-cyano-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridin-6-yl)ethyl]pyridine-3-carboxamide
2-[1-cyclopentyl-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(3-methoxyphenyl)methyl]-N-methylacetamide
1-[2-(2-ethylphenoxy)ethyl]-4-(oxolane-2-carbonyl)piperazine
5-(3-methoxyphenoxymethyl)-N-(quinolin-6-ylmethyl)-1,2-oxazole-3-carboxamide
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N4-(pyridin-4-ylmethyl)-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-1H-1,3-benzodiazole
N-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
N-methyl-5-{[methyl({1H-pyrrolo[2,3-b]pyridin-6-yl})amino]methyl}pyrimidin-2-amine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-(3,4,5-trifluorophenyl)ethan-1-one
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}-N-(2-fluorophenyl)propanamide
6-(azepan-1-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N,N-dimethyl-3-(1-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-3-yl)propanamide
N-[(2-fluorophenyl)methyl]-3-[1-(1,2,4-oxadiazol-3-ylmethyl)piperidin-3-yl]propanamide
1'-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}spiro[indene-1,4'-piperidine]
2-phenyl-N-[1-(pyridin-2-yl)propyl]benzamide
2-cyclopentyl-9-(5-phenyl-1,3,4-thiadiazol-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-cyanopiperidine-1-carbonyl)-N-(1H-imidazol-2-ylmethyl)benzene-1-sulfonamide
8-[2-(4-hydroxyphenyl)acetyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-[(4aS,8aR)-decahydroisoquinoline-2-carbonyl]-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)-1-phenylmethanesulfonamide
7-cyclohexyl-2-(pyridine-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(3-methylpiperidin-1-yl)-3-[2-(1H-1,2,4-triazol-5-yl)benzamido]benzamide
methyl 4-{2-methyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-4-oxobutanoate
1-(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidin-3-yl)pyrrolidin-2-one
1-{4-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}-3,5-dimethyl-1H-pyrazole
3-{[(4-fluorophenyl)methyl]amino}-N-[2-(2-hydroxyethoxy)ethyl]benzamide
8-methyl-2-(1-methyl-1H-pyrazol-4-yl)-4-[4-(pyridin-3-yl)piperazine-1-carbonyl]quinoline
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-N-(2-methylphenyl)piperazine-1-carboxamide