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2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]acetamide
methyl 1-[5-(2-cyclopentylacetamido)-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-4-carboxylate
1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperazine
4-(2,3-difluorobenzoyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-methyl-5-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[4-(propan-2-yloxy)phenyl]methyl}piperazin-2-yl}ethan-1-ol
N-(2-hydroxyethyl)-1-methyl-N-(1,3-thiazol-2-ylmethyl)-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-(methoxymethyl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}cyclobutane-1-carboxamide
4-(5-acetyl-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(2S,4R)-4-amino-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(3-acetamidophenyl)-4-(2,2,2-trifluoroethyl)piperazine-1-carboxamide
(2R)-1-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-2-phenylethan-1-one
N-[(1-benzylpiperidin-4-yl)methyl]-1-[(2-chlorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
(2S,4S,5R)-5-(4-chlorophenyl)-4-[(2-hydroxyethyl)(methyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
3-(methanesulfonylmethyl)-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine
5-(2-fluoro-5-methoxyphenyl)-2,4-dimethoxypyrimidine
(2S,4S)-N,N-diethyl-4-[2-(3-fluorophenoxy)acetamido]-1-methylpyrrolidine-2-carboxamide
1-[(3R,4S)-4-(dimethylamino)-3-(3-hydroxypropyl)piperidin-1-yl]-3-(3,4-dimethylphenyl)propan-1-one
1-({[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}methyl)cyclohexan-1-ol
(9aR)-2-methyl-8-(naphthalene-2-sulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-3-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}urea
2-amino-6-(3,4-dichlorophenyl)-4-(piperidin-3-yl)pyridine-3-carbonitrile
3-[5-(quinoline-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]benzonitrile
(3S,5R)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
N-[(2R,3R)-1'-(3,5-difluorobenzoyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
5-(3-methoxyphenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
(2-{2-[1-(3-chloro-2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
4-(benzyloxy)-1-(oxane-4-carbonyl)piperidine
1-[5-(2H-1,3-benzodioxole-5-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
(1R,5R)-6-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
6-methyl-2-[5-(oxan-2-yl)furan-2-yl]-1H-1,3-benzodiazole
methyl 3-{[2-(4-chloro-2-methylphenoxy)acetamido]methyl}-5-[2-(1H-pyrazol-1-yl)acetamido]benzoate
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-[(2-methoxyphenyl)methyl]cyclopropanamine
2-amino-6-cyclopropyl-4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
1-[7-(1,3-benzothiazol-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
7-methyl-2-phenyl-N-[1-(pyridin-3-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]propyl}piperidine
4-(1-benzothiophen-3-yl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
N-{[1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-3-yl]methyl}acetamide
4-[(3,5-difluorophenyl)methyl]-7-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopropanecarbonyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)piperidine
2,4-dimethyl-N-(1-{4-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)benzamide
N-methyl-5-[(3-methyl-3-phenylpiperidin-1-yl)methyl]-1,2,4-oxadiazole-3-carboxamide
(2S,4S)-4-(2-cyanobenzamido)-N,N-diethyl-1-propanoylpyrrolidine-2-carboxamide
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-3-(1-methylpiperidin-3-yl)propanamide
5-benzyl-4-[3-(dimethylamino)propyl]-1-(2-methylphenyl)piperazin-2-one
7-[(4-fluorophenyl)methyl]-2-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,7-diazaspiro[4.5]decane
1-(4-methyl-1,3-oxazole-5-carbonyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
2-methyl-6-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one