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2-ethyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
2-(3-fluorophenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]azepane
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1,2-dihydrophthalazin-1-one
3-{1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}-N-(4-methoxy-2-methylphenyl)propanamide
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]benzamide
3-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
N-(2-methoxyethyl)-4-methyl-3-[2-oxo-2-(1,2,3,6-tetrahydropyridin-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridine
2-[5-(2,2-dimethylpropyl)-4-phenyl-1H-imidazol-1-yl]-1-(pyridin-3-yl)ethan-1-ol
1-[1-(3-chloro-4-methylphenyl)piperidin-4-yl]-3-(hydroxymethyl)piperidin-3-ol
2-[5-(7-fluoro-2-methylquinolin-4-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
2-(furan-2-yl)-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-oxoacetamide
4-(1-ethylpiperidin-4-yl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
8-[(4-methoxyphenyl)methyl]-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(dimethylamino)-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)acetamide
N-(1-methyl-3-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)piperidine-4-carboxamide
N-{[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}benzamide
N-(furan-2-ylmethyl)-1-methyl-6-oxo-N-(2-phenylethyl)-1,6-dihydropyridazine-3-carboxamide
2-(4-{1-[(3,5-dimethoxyphenyl)methyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)ethan-1-ol
4-(2,3-dihydro-1-benzofuran-7-yl)-N,N-dimethyl-5,6,7,8-tetrahydroquinazolin-2-amine
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine
1-[3-(benzyloxy)phenyl]-3-[(1R,2S)-2-(methoxymethyl)cyclopentyl]urea
1-[1-ethyl-3-(4-phenylpiperazine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-phenylbutan-1-one
3-(4-chlorobenzoyl)-1-(1H-pyrazol-3-ylmethyl)piperidine
4-[(benzylsulfamoyl)amino]-N-ethylpiperidine-1-carboxamide
3-{2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
8-(2,3,6-trimethylquinoline-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[4-(6-aminopyrimidin-4-yl)-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-methyl-N-(2-phenylethyl)piperidine-3-carboxamide
N-benzyl-N-methyl-3-({[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
(3R,4S)-1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,4-dimethylpiperidin-4-ol
3-[2-oxo-2-(3-propanoylpiperidin-1-yl)ethyl]-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidine-2,5-dione
5-(3-methoxyphenyl)-2-(pyridin-4-yl)-4-[1-(thiophen-2-ylmethyl)piperidin-4-yl]pyrimidine
5-benzyl-5-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[(1-ethyl-1H-indazol-3-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
(2S)-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N,3-dimethylbutanamide
methyl (2S,4R)-4-[3-(4-fluorophenyl)benzamido]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carboxylate
2-{[methyl(thiophen-3-ylmethyl)amino]methyl}-4-(pyrimidin-2-yl)phenol
3-{[methyl({[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amino]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1,3-benzothiazol-6-yl)-3-[(3-hydroxypiperidin-1-yl)methyl]benzamide
6-(3,4,5-trimethoxyphenyl)-1H-1,3-benzodiazole
N-(1-methyl-1H-pyrazol-4-yl)-4-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}benzamide
5-[(2-fluoro-4-methoxyphenyl)methyl]-5-{3-oxo-3-[4-(quinazolin-4-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
1-cyclopentyl-N-[5-(morpholin-4-yl)pentyl]-6-oxopiperidine-3-carboxamide
N-[1-(3-methoxyphenyl)-5-oxopyrrolidin-3-yl]-2-methyl-1-benzofuran-5-carboxamide
3,6-dimethyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-1-benzofuran-2-carboxamide