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N-(4,6-dimethylpyridin-2-yl)-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}benzamide
2-(4-{[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(1,3-benzothiazol-2-yl)-3-benzyl-4-methylpiperidin-4-ol
N-methyl-5-{[3-(methylsulfanyl)phenyl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N4-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-5-ethylpyrimidine-2,4-diamine
7-methoxy-2-{4-[3-(methoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
1-(4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)ethan-1-one
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-[(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methylpyrrolidine-3-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-(4-cyclohexanecarbonylpiperazin-1-yl)-2-[(3-fluorophenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(4-fluorophenyl)methyl]-3-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}propanamide
(3S,9aR)-3-(hydroxymethyl)-8-[(3-methoxyphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N,1-dimethyl-N-(oxan-2-ylmethyl)-3-propyl-1H-pyrazole-5-carboxamide
N-{[7-(1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenoxypropanamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(1-propylpiperidin-4-yl)propanamide
methyl 2-({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)-4-(methylsulfanyl)butanoate
({4-ethyl-5-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(2-phenylpropyl)piperidine-4-carboxamide
4-ethyl-3-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(4-benzylpiperidin-1-yl)-1-ethyl-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-{4-[(4-methoxynaphthalen-1-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-[1-(2-{4-[(3-methoxyphenyl)methyl]-3-oxopiperazin-1-yl}-2-oxoethyl)-1H-pyrazol-4-yl]-2-methylfuran-3-carboxamide
2-(4-{[4-(furan-2-yl)phenyl]methyl}-1-(1-methylpiperidin-4-yl)piperazin-2-yl)ethan-1-ol
2-methyl-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1,4-diazepan-5-one
2-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,4S)-2-(2-fluorophenyl)-5-{[4-(methylsulfanyl)phenyl]methyl}-2,5-diazabicyclo[2.2.1]heptan-3-one
5-cyclopropyl-N-[(2S)-oxolan-2-ylmethyl]-1,3-oxazole-4-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,2,6,8-tetramethylquinoline-4-carboxamide
3-[1-(2,6-dimethoxypyridine-3-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
1-[(3,5-dimethylphenyl)methyl]-4-[2-(oxolan-2-ylmethoxy)acetyl]piperazin-2-one
(4S)-3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-4-(propan-2-yl)-1,3-oxazolidin-2-one
(2S,3R)-3-hydroxy-2-({1-[(4-methylphenyl)amino]cyclopentyl}formamido)butanamide
1-[1-(6-methylpyrimidin-4-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
7-{[5-(methoxymethyl)furan-2-yl]methyl}-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
4-(2-methylphenoxy)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-(3-methylbutyl)-1H-pyrazole-4-carboxamide
4-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-N-methylpyridin-2-amine
2-(5-{1-[2-hydroxy-5-(1H-pyrrol-1-yl)benzoyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetic acid
N-methyl-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-2-(methylamino)-1,3-thiazole-4-carboxamide
2-[4-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-chloro-N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(3-methylpentanoyl)piperidin-4-yl]imidazolidine-2,4-dione
3-[(3-{4-[3-(trifluoromethyl)phenyl]-1H-pyrazol-5-yl}piperidin-1-yl)methyl]pyridine
4-{3-methyl-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}benzene-1-sulfonamide
N-[(3S,4R)-1-[(2,4-dichlorophenyl)methyl]-4-propylpyrrolidin-3-yl]acetamide
N-methyl-N-{2-[(5-methylhex-5-en-2-yl)amino]ethyl}methanesulfonamide
5-{4-[1-(N-methyl-1-pyridin-2-ylformamido)-2-phenylethyl]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate