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1-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydroquinolin-2-one
5-{3-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-oxopropyl}-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
[(3R,4R)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-(3-fluorophenyl)-4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-2-one
N-[(3-phenylphenyl)methyl]morpholine-2-carboxamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,2-dimethylpropanamide
2-(4-chloro-2-methylphenoxy)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
5-ethyl-5-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
(3S,4R)-1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(hydroxymethyl)piperidin-3-ol
5-fluoro-2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N-methyl-N-[3-(piperidin-1-yl)propyl]-1H-1,3-benzodiazole-7-carboxamide
2-[5-(5-ethyl-2-methylpyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-(2-chloro-6-methylphenyl)-4-[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
3-(carbamoylamino)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
2-(3-fluorophenyl)-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N,N-dimethyl-7-(oxolane-3-carbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-benzyl-3-ethyl-1-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-5-one
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
3-{[4-(4H-1,2,4-triazol-4-yl)piperidin-1-yl]methyl}phenol
2-{2-[3-(pyrrolidine-1-carbonyl)phenyl]phenoxy}propanamide
5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
[3-(2-methylquinolin-5-yl)phenyl]methanamine
(3S,4S)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-propylpyrrolidine-3-carboxylic acid
3-(2,3-dihydro-1H-inden-2-yl)-5-[1-(2-methoxypyridine-3-carbonyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-(phenoxymethyl)-1H-1,3-benzodiazole
5-{1-[2-(cyclohex-1-en-1-yl)acetyl]pyrrolidin-2-yl}-N-(pyridin-2-yl)thiophene-2-carboxamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-6,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
1-(3-methylpyridin-2-yl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(3-methylbutyl)piperidin-4-ol
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-3-acetamidopropanamide
1-(4-chloro-3-methylbenzoyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}-N-(furan-2-ylmethyl)acetamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydro-1-benzofuran-2-carboxamide
N-[(8-{[3-(trifluoromethyl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]oxolane-2-carboxamide
2-(1H-imidazol-2-yl)-N-[3-(4-methylpiperazin-1-yl)propyl]benzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-ethyl-5-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
6-methyl-2-oxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
3-[2-(2-hydroxyphenyl)ethyl]-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(pyridin-4-yl)-1-(thiophen-3-ylmethyl)pyrrolidine-3-carboxylic acid
5-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(1R,9aR)-1-(3-benzyl-1H-1,2,4-triazol-5-yl)-octahydro-1H-quinolizine
5-(3-fluorophenoxymethyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-3-carboxamide
[(3R,4S)-1-{[3-(morpholin-4-yl)phenyl]methyl}-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
4-(1-methylpiperidin-4-yl)-1-[2-(pyrrolidin-1-yl)benzoyl]piperidine
N-({7-[2-(2,3-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(methylsulfanyl)benzamide
1-(2-cyclohexylethyl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(dimethylamino)ethyl]-5-{thieno[3,2-d]pyrimidin-4-yl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide