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1-(oxolan-2-ylmethyl)-N-(1-phenylcyclopropyl)-1H-1,2,3-triazole-4-carboxamide
[(3-{2-[1-(2-fluorobenzoyl)piperidin-2-yl]ethoxy}phenyl)methyl](methyl)(quinolin-8-ylmethyl)amine
3-(5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)propanoic acid
1-[1-(4-fluorophenyl)ethyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
methyl 4-{5-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]-1,2,4-oxadiazol-3-yl}benzoate
N-[2-(2,4-difluorophenyl)-1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}quinoline
2-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazine-1-carbonyl)-7-fluoro-3-methyl-1H-indole
(3S,4R)-4-(3-methylthiophen-2-yl)-1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperidin-3-ol
methyl 3-[2-(1H-pyrazol-1-yl)acetamido]-5-({[3-(trifluoromethyl)phenyl]formamido}methyl)benzoate
methyl 2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl}-6-[(2E)-4-methylpent-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
N-(3-chloro-2-propoxyphenyl)-2-(2-methoxyethyl)morpholine-4-carboxamide
N-[5-(cyclopropylcarbamoyl)-2-methoxyphenyl]-2-methyl-3-oxopiperazine-1-carboxamide
1-[4-(4-ethoxy-3-methylphenyl)butanoyl]-N-methylpyrrolidine-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-methylpyrimidin-4-yl)pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
2-(2-{[2-(2,3-dimethylphenoxy)ethyl]amino}ethyl)-1,2-dihydrophthalazin-1-one
2-{5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
methyl (2S)-1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
{1-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]piperidin-4-yl}methanol
5-{[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]methyl}-3-(phenoxymethyl)-1,2,4-oxadiazole
1-[(4-fluorophenyl)methyl]-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
6-({[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}methyl)-1,4-oxazepan-6-ol
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3,5-dimethoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-fluorophenyl)methyl]-4-(3-fluoropyridine-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
S-(2-acetyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-hydroxybutane-1-sulfonamido
methyl 3-[(4-fluoro-3-methoxyphenyl)methyl]-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[2-(thiophen-2-yl)ethyl]propanamide
N-[(3R,4S)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-phenylpyrrolidin-3-yl]cyclobutanecarboxamide
6-methyl-14-(3-methyl-1H-pyrazol-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
methyl 5-{[(3,5-dimethylphenyl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-[(1S,5R)-6-(5-methoxyfuran-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
3-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(4-sulfamoylphenyl)urea
N-[(3-chlorophenyl)methyl]-5-hydroxy-N-propylpyrazine-2-carboxamide
N-{2-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-methoxypropanamide
8-(5-acetylpyridin-2-yl)-2-benzyl-2,8-diazaspiro[4.5]decan-3-one
1-[4-(3-fluorophenyl)phenyl]-N-[2-(1H-pyrazol-1-yl)ethyl]piperidin-4-amine
N-[(2R,3R)-2-hydroxy-1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methoxybenzamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
2-[2-oxo-2-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
N-[3-(cyclohexylsulfanyl)propyl]-2-methyl-1,3-thiazole-4-carboxamide
N-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropanamine
2-(4-methylpentanoyl)-7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-6-one
3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
4-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
2-amino-6-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrimidine-4-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2S)-1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]acetamide