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2-butyl-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidine
1-(methoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]cyclobutane-1-carboxamide
6-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-methyl-2,3-dihydropyridazin-3-one
(1R,5S,6S)-6-{[4-(1,3-thiazol-2-yl)piperazin-1-yl]methyl}-3-azabicyclo[3.1.0]hexane
5-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-(2-chlorophenyl)-N-{[8-(pyridine-4-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
6-(2,5-dimethylphenyl)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(4aR,7aS)-1-methyl-4-(7-methyl-1-benzofuran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-fluoro-N-(2-methoxyethyl)-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-[({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
(2S)-3-(4-hydroxyphenyl)-2-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]propanoic acid
ethyl 2-[3-(2H-1,3-benzodioxol-5-yl)-N-methyl-3-phenylpropanamido]acetate
1-{2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxybenzoyl}piperidin-4-ol
methyl 3-{[5-(2-chlorobenzoyl)-1-(cyclopropylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
6-(cyclopentylmethyl)-2-[3-(1,4-oxazepan-4-ylmethyl)phenyl]-3,4-dihydropyrimidin-4-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-(1-methylcyclopropyl)-N-(oxolan-2-ylmethyl)propanamide
2-(1'-{2-[(cyclopropylmethyl)sulfanyl]acetyl}-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl)acetamide
(3R,5R)-N-methyl-5-(morpholine-4-carbonyl)-N-(quinoxalin-2-ylmethyl)piperidine-3-carboxamide
4-cyclopentyl-N-(1-methyl-1H-1,3-benzodiazol-5-yl)-3-oxopiperazine-1-carboxamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(4-fluorophenyl)ethyl]propanamide
1-(furan-2-ylmethyl)-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]methanol
(1R,5R)-6-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-[1-(2-methoxyacetyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
N-ethyl-4-[2-(1H-pyrazol-1-yl)butanamido]piperidine-1-carboxamide
[(3R,4R)-1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carbonyl]-1-(2-methylpropyl)pyrrolidin-2-one
4-(2-methyl-1H-imidazol-1-yl)-1-(quinolin-4-yl)piperidine-4-carboxylic acid
N-(1,4-dioxan-2-ylmethyl)-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
1-{[1-(1-benzothiophene-5-carbonyl)piperidin-4-yl]methyl}pyrrolidin-2-one
N-methyl-N-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(8-methoxyquinolin-5-yl)methyl](methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(furan-2-ylmethyl)(isoquinolin-5-ylmethyl)(thiophen-3-ylmethyl)amine
N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-(thiophen-2-yl)butanamide
1-(1H-indazol-7-yl)-3-methyl-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}urea
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-6-methoxypyrimidin-2-amine
2-[3-(1H-pyrazol-3-yl)phenyl]-6-(trifluoromethyl)pyridine
4-[5-(3-ethynylbenzoyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]piperazin-2-one
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
2-{4-cyclobutyl-1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-4-({[3-(dimethyl-1,2-oxazol-4-yl)propyl]carbamoyl}amino)benzamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}propanamide
5-(2-methoxyacetamido)-1-methyl-N-[2-(propan-2-yloxy)ethyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-1-[(4-methoxyphenyl)methyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(3S)-1,3-dimethyl-4-(3-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazin-2-one
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(trifluoromethyl)piperidine
1-[4-(furan-2-yl)benzoyl]-4-[(3-methylpyridin-2-yl)methyl]piperazine
methyl 4-[(2R,3R)-2-(2-methoxyethoxy)-3-propanamido-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-ylmethyl]benzoate