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[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
N-ethyl-5-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)pyrimidin-2-amine
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(2-ethylphenoxy)azetidine
2-(3-methylthiophen-2-yl)-1-(oxan-3-ylmethyl)-1H-imidazole
2-(pyridin-3-yl)-N-[1-(thiophen-2-yl)butyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)cyclobutanecarboxamide
6-(2-chlorophenyl)-N-cyclobutylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-{1-[1-(2,4-difluorobenzoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
N-methyl-5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-N-(pyrimidin-4-ylmethyl)pyridin-2-amine
ethyl 1-[(3-methoxyphenyl)methyl]-5-(2-methylpropanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
3-cyclopropaneamido-4-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]benzamide
1-{1-[6-(2,3-dimethylphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[2-(3-{[methyl(thiophen-2-ylmethyl)amino]methyl}phenoxy)ethyl]piperazin-1-yl}ethan-1-one
5-fluoro-2-methyl-N-[(3S)-2-oxoazepan-3-yl]-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
5-propyl-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-(2-methyl-1,3-benzothiazol-5-yl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
N-[(4-phenyl-1,3-thiazol-5-yl)methyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
2-(2,5-dimethoxyphenyl)-3-methylquinoxaline
2-methoxy-2-phenyl-N-{1-[1-(propan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
methyl 3-[cyclopropyl({[3-(oxolan-3-ylmethoxy)phenyl]methyl})sulfamoyl]thiophene-2-carboxylate
2-oxo-1-(2-phenylethyl)-3-(pyridin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
3-[(2-methoxyethyl)sulfamoyl]-5-(4-methoxyphenyl)benzoic acid
2-methoxy-N-(3-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}phenyl)benzamide
N-(1-{7-[(3,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylbenzamide
({2,5-dimethyl-3-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
4-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[(1r,4r)-4-methylcyclohexanecarbonyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(4-chlorophenyl)-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}cyclobutane-1-carboxamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-[(2-methoxyphenyl)methyl]acetamide
4-(2,5-dimethoxyphenyl)-2-({4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}methyl)phenol
[(3R,4S)-1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(3-ethyl-1H-pyrazole-5-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
3-(1-butyl-1H-imidazol-2-yl)-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidine
N,N-diethyl-7,8-dimethyl-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
(4aS,7aR)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpropanamide
N-benzyl-N-methyl-1-[2-(pent-4-enamido)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-1,3-oxazole-4-carboxamide
8-(morpholine-2-carbonyl)-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-{[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]sulfonyl}benzonitrile
3-(4-fluorophenoxymethyl)-1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidine
2-(methylsulfanyl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}pyridine-3-carboxamide
4-{[1-(cyclopent-1-ene-1-carbonyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
5-methoxy-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]furan-2-carboxamide
2-(4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrimidine
5-[(3-{4-[(2-fluorophenyl)methyl]piperidine-1-carbonyl}-1,2-oxazol-5-yl)methoxy]isoquinoline
1-(4-hydroxy-4-phenylpiperidin-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
(4S)-4-[3-(3,4-difluorophenyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-4-acetamidobutanamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-methyl-3-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]urea