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[7-(6,8-dimethoxy-4-methylquinolin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methanamine
N-(3-hydroxyadamantan-1-yl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
4-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
1-[2-(3-phenylpropyl)morpholin-4-yl]-2-(pyridin-4-yl)ethan-1-one
1-[(4-ethoxyphenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-4-phenylbutane-1,4-dione
N,2,5,6-tetramethyl-N-[4-(morpholin-4-yl)butyl]pyrimidin-4-amine
N-[2-(2-chlorophenyl)ethyl]-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
2-methyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]thieno[3,2-d]pyrimidin-4-amine
2-[1-(7-fluoro-3-methyl-1-benzofuran-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-[3-(4-methylphenoxy)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-chloro-2-fluoro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
methyl 3-({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}carbamoyl)propanoate
2-[1-(3-methylbutyl)-8-{[3-(2-methylphenyl)phenyl]methyl}-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
methyl 6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-phenoxyacetamide
[(8-chloroquinolin-2-yl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
5-(naphthalen-2-yl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2,4-triazin-3-amine
1-{2-[3-methyl-4-({[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1H-pyrazol-1-yl]ethyl}piperidin-4-ol
2-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(1-cyclobutanecarbonylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
2-[(3,4-difluorophenyl)methyl]-8-[(2E)-2-methylbut-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
(2,1,3-benzoxadiazol-5-ylmethyl)({5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)methylamine
3-[({1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}oxy)methyl]pyridine
2-(2,5-dimethoxyphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-cyclopropylacetamide
(1R,2S,9R)-11-(2,3-dihydro-1-benzofuran-5-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N,N-bis(prop-2-en-1-yl)-1H-1,3-benzodiazole-7-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-3,4,5-trimethoxy-N-(oxolan-2-ylmethyl)benzamide
4-[4-(1-phenyl-1H-imidazol-4-yl)benzoyl]piperazine-2-carboxylic acid
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
2,2-dimethyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)oxane-4-carboxamide
dimethyl({[(1R,5S,6S)-3-[3-(1H-pyrazol-1-yl)benzoyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-butyl-1-methyl-4-[4-(2-methylpropyl)benzoyl]piperazin-2-one
N,N-dimethyl-2-{methyl[2-methyl-2-(morpholin-4-yl)propyl]amino}propanamide
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
(3S)-N-tert-butyl-2-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-(1-{7-[(2E)-2-methylbut-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
N-methyl-2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
3-methyl-N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}methyl)-1H-pyrazole-5-carboxamide
N-cyclopropyl-2-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-4-carboxamide
4-{[(5-{1-[(3,4-difluorophenyl)methyl]-1H-pyrazol-3-yl}furan-2-yl)methyl]amino}-1-methylpyrrolidin-2-one
(2S,4S,5R)-4-{[2-(1H-imidazol-1-yl)ethyl]carbamoyl}-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
2-ethyl-N-{[4-(3-methoxyphenyl)-5-({[3-(trifluoromethyl)phenyl]methyl}sulfanyl)-4H-1,2,4-triazol-3-yl]methyl}butanamide
1-[(3-methoxyphenyl)methyl]-4-(5-phenyl-1,2,4-oxadiazol-3-yl)piperazin-2-one
methyl 3-(cyclopropylmethyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2,2-dimethylpropan-1-one