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1-[4-(pyridin-3-yloxy)piperidin-1-yl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
N-(3-ethoxypropyl)-1-methyl-3-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 1-{[1-(cyclobutylmethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}piperidine-4-carboxylate
3-cyclopropyl-5-[(2-propyl-1H-imidazol-1-yl)methyl]-1,2,4-oxadiazole
{[7-(azocane-1-carbonyl)-1-methyl-2-(2-methylpropyl)-1H-1,3-benzodiazol-5-yl]sulfamoyl}dimethylamine
N,N-diethyl-4-{3-[(2-phenylethyl)carbamoyl]piperidin-1-yl}piperidine-1-carboxamide
2-(5-fluoro-2-methylphenyl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
methyl 3-[4-({8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}methyl)-1H-pyrazol-1-yl]propanoate
N-(2-hydroxyethyl)-5-(methoxymethyl)-N-[(3-methylthiophen-2-yl)methyl]thiophene-2-carboxamide
(1S,5R)-3-(5-chloro-2-methoxybenzoyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[1-(cyclohexylmethyl)-1H-pyrazol-4-yl]-1-methyl-1,2,3,6-tetrahydropyridine
2-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrazol-4-yl}ethan-1-ol
4-methyl-3-[2-methyl-3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
5-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
N-cyclopropyl-1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-methyl-2-(4H-1,2,4-triazol-4-yl)-5-(2,3,4-trimethoxyphenyl)pyridine
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}imidazolidine-2,4-dione
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-ethyl-1,4-diazepan-5-one
2-(4-{[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]methyl}phenyl)acetic acid
3-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}-1,3-oxazolidin-2-one
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
4-methoxy-N-{[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-[(1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}piperidin-4-yl)methyl]acetamide
7-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N,N-dimethyl-2,7-diazaspiro[4.5]decane-2-carboxamide
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methyl-1H-imidazol-4-yl)methyl]piperidine
1-cyclohexyl-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-ethylpyrimidine-5-carboxamide
2-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
(3aS,6aS)-2-cyclobutanecarbonyl-5-(4-ethyl-5-methylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-benzyl-2-(1-benzyl-3-oxopiperazin-2-yl)-N-(cyclopropylmethyl)acetamide
N-[2-(2-chlorophenyl)ethyl]-1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
3-{[1-(3-ethoxypropanoyl)pyrrolidin-3-yl]methyl}benzoic acid
3,3,3-trifluoro-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
[3-(cyclopropylmethyl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]piperidin-3-yl]methanol
(4-{4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}pyridin-2-yl)methanol
4-(3,4,5-trimethoxyphenyl)benzamide
2-(5-{2H,3H-thieno[3,4-b][1,4]dioxin-5-yl}-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl)acetic acid
2-(1-ethyl-5-methyl-1H-pyrazol-4-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
1-[3-(4-fluorophenyl)-5-[2-(4-methylpiperazin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
N-[2-(furan-2-yl)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
2-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(thiophen-3-yl)acetic acid
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2,4-dimethyl-N-(1-{4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]phenyl}-1H-pyrazol-4-yl)benzamide
4-methyl-3-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]benzamide
3-[({2-[(4-chlorophenyl)methoxy]ethyl}amino)methyl]piperidin-3-ol
2-methyl-2-[(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)formamido]propanamide
methyl 1-(3-{3-[(tert-butylamino)methyl]phenoxy}-2-hydroxypropyl)piperidine-4-carboxylate
N-methyl-3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyridin-2-amine