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3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[1-(pyrazin-2-yl)propan-2-yl]urea
(4aR,8aS)-6-(1H-indol-2-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
N-(1-{4-[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]phenyl}-1H-pyrazol-4-yl)furan-3-carboxamide
2-(2-aminoethyl)-5,6-dimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]thieno[2,3-d]pyrimidin-4-amine
5-{5-methylthieno[2,3-d]pyrimidin-4-yl}quinoline
N-[(2-chlorophenyl)methyl]-7-cyclobutaneamido-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
methyl 1-(benzyloxy)-2-oxo-8-(quinolin-4-ylmethyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
3-(4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)pyridine
3-[5-(1H-pyrrole-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-(3-fluoro-4-methoxybenzoyl)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
4-(1H-pyrazol-1-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}benzene-1-sulfonamide
methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})(oxolan-3-ylmethyl)amine
1-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-4-(piperidin-1-yl)butan-1-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-phenyl-1,2,4-triazin-3-amine
N-methyl-4-({4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}sulfonyl)thiophene-2-carboxamide
4'-(1,4-dioxan-2-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[2-methoxy-4-({[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-(thiophen-3-yl)-5-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2,4-oxadiazole
5-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}-N,N-dimethyl-1,3-thiazol-2-amine
2-[4-(1-benzofuran-2-sulfonyl)morpholin-3-yl]acetic acid
1-methyl-4-phenyl-3-{[1-(pyrimidine-4-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-N,N-dimethylpyrrolidin-3-amine
1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-(2-fluorophenoxy)piperidine
N-{[7-(3,3-dimethylbutanoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}thiophene-2-sulfonamide
2-({4-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)morpholine
methyl 4-[5-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
5-[1-(2,3-dimethylbenzoyl)piperidin-4-yl]-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-[4-(3-methyl-2-oxoimidazolidin-1-yl)phenyl]urea
5-methyl-3-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
6-methyl-N4-{[4-(methylsulfanyl)phenyl]methyl}pyrimidine-2,4-diamine
4-(dimethyl-1,2-oxazol-4-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(3,4-dimethylphenyl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-amine
(2R,6R)-4-(2,3-dimethoxybenzoyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N'-(4-methylphenyl)-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]propanediamide
9-methoxy-4-[(3-methylphenyl)methyl]-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,8aR)-1-(4-hydroxybutyl)-6-(morpholine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 1-[(3,4-dimethoxyphenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[(3S,4R)-1-[2-(5-acetylthiophen-3-yl)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-(furan-2-yl)-N-[2-(1H-1,2,3-triazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N,N-dimethyl-7-(1-phenylcyclopropanecarbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3aR,6aR)-2-cyclopentanecarbonyl-5-(5-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-({5-phenylmethanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2,5-dihydro-1H-pyrrole
3-{3-ethyl-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
2,6-dimethoxy-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}pyridine-3-carboxamide
4-(2-methoxyethoxy)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(1-methoxybutan-2-yl)amino]piperidin-1-yl}benzamide
(2S,4S)-4-amino-1-{[2-(benzyloxy)phenyl]methyl}-N-ethylpyrrolidine-2-carboxamide